Novel Catalyst System for Suzuki-Miyaura Coupling of Challenging DNA-Linked Aryl Chlorides

Bioconjug Chem. 2016 Nov 16;27(11):2597-2600. doi: 10.1021/acs.bioconjchem.6b00541. Epub 2016 Oct 12.

Abstract

A novel Pd catalyst system, [(t-Bu)2P(OH)]2PdCl2 (POPd) with the ligand sodium 2'-(dicyclohexylphosphino)-2,6-dimethoxy-[1,1'-biphenyl]-3-sulfonate, is reported. It effectively catalyzes the Suzuki-Miyaura coupling of challenging phenyl chlorides and pyrimidinyl chlorides that are covalently linked to a double-stranded DNA-template with various boronic acids/esters.

MeSH terms

  • Catalysis
  • Chlorides / chemistry*
  • DNA / chemistry*
  • Ligands
  • Models, Molecular
  • Nucleic Acid Conformation
  • Palladium / chemistry*

Substances

  • Chlorides
  • Ligands
  • Palladium
  • DNA