Ibuprofen loaded PVA/chitosan membranes: A highly efficient strategy towards an improved skin wound healing

Carbohydr Polym. 2017 Mar 1:159:136-145. doi: 10.1016/j.carbpol.2016.12.029. Epub 2016 Dec 13.

Abstract

During wound healing, an early inflammation can cause an increase of the wound size and the healing process can be considerably belated if a disproportionate inflammatory response occurs. (S)-ibuprofen (IBP), a non-steroidal anti-inflammatory agent, has been used for muscle healing and to treat venous leg ulcers, but its effect in skin wound healing has not been thoroughly studied thus far. Herein, IBP-β-cyclodextrins carriers were designed to customise the release profile of IBP from poly(vinyl alcohol)/chitosan (PVA/CS) dressings in order to promote a faster skin regeneration. The dressings were produced using supercritical carbon dioxide (scCO2)-assisted technique. In vitro IBP release studies showed that β-cyclodextrins allowed a controlled drug release from the hydrogels which is crucial for their application in wound management. Moreover, the in vivo assays revealed that the presence of PVA/CS membranes containing IBP-β-cyclodextrins carriers avoided scab formation and an excessive inflammation, enabling an earlier skin healing.

Keywords: Composite membranes; Drug delivery systems; Ibuprofen; In vivo assays; Supercritical carbon dioxide; Wound dressings.

MeSH terms

  • Animals
  • Bandages / standards
  • Cells, Cultured
  • Chitosan / chemistry*
  • Female
  • Humans
  • Ibuprofen / chemistry*
  • Polyvinyl Alcohol / chemistry
  • Rats
  • Rats, Wistar
  • Skin / injuries*
  • Wound Healing*

Substances

  • Polyvinyl Alcohol
  • Chitosan
  • Ibuprofen