Trimethylamine N-oxide promotes atherosclerosis via CD36-dependent MAPK/JNK pathway

Biomed Pharmacother. 2018 Jan:97:941-947. doi: 10.1016/j.biopha.2017.11.016. Epub 2017 Nov 7.

Abstract

Background: Many studies have identified trimethylamine N-oxide (TMAO) as a new risk factor of cardiovascular diseases. It has been suggested that TMAO promotes atherosclerosis development. However, the underlying mechanism is still unclear.

Methods: Apoe-/- mice were fed a high-fat diet and given water with or without TMAO for 8-week. Histological and immunohistological analyses were used to evaluate the atherogenic effect of TMAO in vivo. We also employed peritoneal elicited macrophages and RAW264.7 to assess the role of MAPK/JNK pathway in TMAO-induced formation of foam cells.

Results: TMAO significantly promoted plaque progression in apoe-/- mice fed with high-fat diet for 8 weeks. Besides, macrophage recruitment, CD36 and proinflammatory cytokine expressions were enhanced by TMAO in plaque lesions. In vitro, TMAO increased the macrophage migration and the expression of TNF-α, IL-6 and ICAM1. In addition, CD36 expression and foam cell formation induced by ox-LDL were also enhanced by TMAO, which could be attenuated by siRNA-mediated knockdown of CD36. We additionally used MAPK inhibitor (SB230580) and JNK inhibitor (SP600125) to assess the MAPK/JNK pathway in TMAO-induced CD36 expression. Western blotting showed that both SB230580 and SP600125 could reduce the expression of CD36 induced by ox-LDL and TMAO. Moreover, SB230580 and SP600125 could also reduce the formation of foam cells.

Conclusions: TMAO promotes the atherosclerosis in vivo and in vitro.CD36/MAPK/JNK pathway may play a crucial role in TMAO-induced formation of foam cells.

Keywords: Atherosclerosis; CD36; Foam cell; Macrophage; TMAO.

MeSH terms

  • Animals
  • Apolipoproteins E / genetics
  • Atherosclerosis / chemically induced*
  • Atherosclerosis / pathology
  • CD36 Antigens / genetics
  • CD36 Antigens / metabolism*
  • Cytokines / metabolism
  • Disease Models, Animal
  • Disease Progression
  • Foam Cells / drug effects
  • Foam Cells / metabolism
  • Gene Knockdown Techniques
  • Lipoproteins, LDL / metabolism
  • MAP Kinase Signaling System / drug effects
  • Macrophages / drug effects
  • Macrophages / metabolism
  • Macrophages, Peritoneal / drug effects
  • Macrophages, Peritoneal / metabolism
  • Male
  • Methylamines / toxicity*
  • Mice
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Plaque, Atherosclerotic / chemically induced*
  • Plaque, Atherosclerotic / pathology
  • RAW 264.7 Cells

Substances

  • Apolipoproteins E
  • CD36 Antigens
  • Cytokines
  • Lipoproteins, LDL
  • Methylamines
  • oxidized low density lipoprotein
  • trimethyloxamine