The chemokine receptor type 4 antagonist, AMD3100, interrupts experimental tooth movement in rats

Arch Oral Biol. 2018 Feb:86:35-39. doi: 10.1016/j.archoralbio.2017.11.003. Epub 2017 Nov 11.

Abstract

Objective: The aim of this study was to clarify the role of the stromal cell-derived factor-1 (SDF-1)/C-X-C chemokine receptor type 4 (CXCR4) axis in osteoclast accumulation, and the influence of orthodontic tooth movement (OTM) under mechanical force application to periodontal tissues, by administration of the CXCR4 antagonist AMD3100.

Design: The upper right first molar (M1) of rats was moved mesially with a 10-g force titanium-nickel closed coil spring. Rats were treated with phosphate-buffered saline or AMD3100 (5mg/kg), which is a SDF-1 antagonist. After 0, 1, 3, and 7days, alveolar bones in all groups were examined at each time point by micro-computed tomography and histological analysis.

Results: Tooth movement was decreased significantly in the AMD3100-treated group at 1, 3, and 7days after beginning OTM. The numbers of tartrate-resistant acid phosphatase-positive multinucleated cells in the periodontal ligament around the maxillary M1 were decreased significantly in the treated as compared to the control group on Days 1 and 3.

Conclusion: Administration of AMD3100 decreases OTM and osteoclast accumulation in rat molars under orthodontic force application. These findings suggest that the SDF-1/CXCR4 axis plays an important role in alveolar bone metabolism during OTM.

Keywords: AMD3100; Orthodontic tooth movement; Osteoclast; Periodontal ligament; Stromal cell-derived factor-1.

MeSH terms

  • Alveolar Process / metabolism
  • Animals
  • Benzylamines
  • Chemokine CXCL12 / antagonists & inhibitors
  • Cyclams
  • Heterocyclic Compounds / pharmacology*
  • Molar
  • Osteoclasts / drug effects
  • Periodontal Ligament / cytology
  • Rats
  • Receptors, CXCR4 / antagonists & inhibitors
  • Tooth Movement Techniques / methods*
  • X-Ray Microtomography

Substances

  • Benzylamines
  • CXCL12 protein, rat
  • Chemokine CXCL12
  • Cxcr4 protein, rat
  • Cyclams
  • Heterocyclic Compounds
  • Receptors, CXCR4
  • plerixafor