Neuroprotective evidence of alpha-lipoic acid and desvenlafaxine on memory deficit in a neuroendocrine model of depression

Naunyn Schmiedebergs Arch Pharmacol. 2018 Aug;391(8):803-817. doi: 10.1007/s00210-018-1509-1. Epub 2018 May 7.

Abstract

Cognitive impairment is present in patients with depression. We hypothesized that alpha-lipoic acid (ALA) can reduce cognitive impairment, especially when combined to antidepressants. Female mice received vehicle or corticosterone (CORT) 20 mg/kg, s.c. for 14 days. From the 15th to 21st day, the animals were divided in groups: vehicle, CORT, CORT+desvenlafaxine (DVS) 10 or 20 mg/kg, ALA 100 or 200 mg/kg, DVS10+ALA100, DVS20+ALA100, DVS10+ALA200, or DVS20+ALA200. Tail suspension (TST), social interaction (SIT), novel object recognition (NOR), and Y-maze tests were conducted. Acetylcholinesterase activity (AChE) was measured in the prefrontal cortex (PFC), hippocampus (HC), and striatum (ST). CORT caused depressive-like behavior, impairment in SIT, and cognitive deficits. Alpha-lipoic acid and DVS, alone or combined, reversed CORT effect on TST. In the NOR, ALA200 alone, DVS10+ALA100, or DVS10+ALA200 reversed the deficits in short-term memory, while DVS20 alone or DVS20+ALA200 reversed the deficits in long-term memory. In the Y-maze test, ALA200 alone, DVS20+ALA100, or DVS20+ALA200 reversed the deficits caused by CORT in the working memory. CORT increased AChE in the PFC, HC, and ST. ALA200 alone or DVS20+ALA200 reversed this effect in the PFC, while DVS20 or DVS20+ALA100 reversed this effect in the HC. In the ST, DVS10 or 20, alone or combined, and ALA100 reversed the effects of CORT. These results suggest that DVS+ALA, by reversing CORT-induced memory and social deficits, seems to be a promising therapy for the treatment of depression and reversal of cognitive impairment observed in this disorder.

Keywords: Acetylcholinesterase; Alpha-lipoic acid; Cognitive impairment; Corticosterone model of depression; Desvenlafaxine; Major depressive disorder.

MeSH terms

  • Acetylcholinesterase / metabolism
  • Animals
  • Antidepressive Agents / therapeutic use*
  • Behavior, Animal / drug effects
  • Brain / drug effects
  • Brain / enzymology
  • Corticosterone
  • Depression / chemically induced
  • Depression / drug therapy*
  • Desvenlafaxine Succinate / therapeutic use*
  • Drug Synergism
  • Female
  • Memory Disorders / chemically induced
  • Memory Disorders / drug therapy*
  • Memory, Short-Term / drug effects
  • Mice
  • Neuroprotective Agents / therapeutic use*
  • Social Behavior
  • Thioctic Acid / therapeutic use*

Substances

  • Antidepressive Agents
  • Neuroprotective Agents
  • Thioctic Acid
  • Acetylcholinesterase
  • Corticosterone
  • Desvenlafaxine Succinate