Tyrosine kinase activity of brain insulin and IGF-1 receptors

Biochem Biophys Res Commun. 1986 Jan 29;134(2):532-8. doi: 10.1016/s0006-291x(86)80453-3.

Abstract

Lectin-purified rat brain preparations demonstrate specific [125I]insulin and [125I]-IGF-1 binding. Insulin-stimulable tyrosine kinase activity as measured by exogenous substrate phosphorylation was present in brain and liver lectin purified preparations with the delta kinase activity/B/F of brain approximately 2.5 fold greater than that of liver. Insulin-stimulable tyrosine kinase activity was abolished in liver but decreased by only approximately 50 percent in brain after immuno-depletion with antiserum which recognizes insulin but not IGF-1 receptors. Insulin and IGF-1 dose responses for phosphorylation of the immunodepleted brain preparations suggested that the remaining tyrosine kinase activity was IGF-1 receptor mediated. Thus, functional IGF-1 receptors are present in rat brain, and the doses of insulin typically used to evaluate insulin receptor tyrosine kinase activity will stimulate IGF-1 receptor tyrosine kinase activity as well.

MeSH terms

  • Animals
  • Brain / enzymology*
  • Insulin-Like Growth Factor I / metabolism*
  • Lectins
  • Liver / enzymology
  • Male
  • Phosphoproteins / metabolism
  • Phosphorylation
  • Protein-Tyrosine Kinases / metabolism*
  • Rats
  • Receptor, Insulin / isolation & purification
  • Receptor, Insulin / metabolism*
  • Receptors, Cell Surface / isolation & purification
  • Receptors, Cell Surface / metabolism*
  • Receptors, Somatomedin
  • Somatomedins / metabolism*

Substances

  • Lectins
  • Phosphoproteins
  • Receptors, Cell Surface
  • Receptors, Somatomedin
  • Somatomedins
  • Insulin-Like Growth Factor I
  • Protein-Tyrosine Kinases
  • Receptor, Insulin