Interaction of clavulanic acid, sulbactam and cephamycin antibiotics with beta-lactamases

Drugs Exp Clin Res. 1987;13(3):145-8.

Abstract

The inhibitory effects of clavulanic acid, sulbactam and cephamycin antibiotics on chromosomally-mediated or plasmid-mediated beta-lactamases were investigated. The inhibition constants were determined by a non-linear regression analysis. Clavulanic acid and sulbactam had high affinities for the purified plasmid-mediated beta-lactamases such as SHV-1, TEM-1 and PSE-4, and were potent inhibitors as shown by their low Ki values. Except for Bacteroides beta-lactamase, which is sensitive to inhibition by cephamycin antibiotics, clavulanic acid and sulbactam were found not to be as effective against chromosomally-mediated beta-lactamases. The cephamycin antibiotics were better inhibitors of chromosomally-mediated beta-lactamases than those that are plasmid mediated. Except for P99 beta-lactamase, against which sulbactam and clavulanic acid were inactive, the cephamycin antibiotics were less effective inhibitors than sulbactam and clavulanic acid.

MeSH terms

  • Anti-Bacterial Agents / pharmacology*
  • Bacteria / drug effects*
  • Bacteria / enzymology
  • Cephamycins / pharmacology*
  • Clavulanic Acid
  • Clavulanic Acids / pharmacology*
  • Drug Interactions
  • Microbial Sensitivity Tests
  • Penicillanic Acid / pharmacology*
  • Sulbactam
  • beta-Lactamase Inhibitors*
  • beta-Lactamases / isolation & purification

Substances

  • Anti-Bacterial Agents
  • Cephamycins
  • Clavulanic Acids
  • beta-Lactamase Inhibitors
  • Clavulanic Acid
  • Penicillanic Acid
  • beta-Lactamases
  • Sulbactam