DNA polymerase ι is acetylated in response to SN2 alkylating agents

Sci Rep. 2019 Mar 18;9(1):4789. doi: 10.1038/s41598-019-41249-3.

Abstract

DNA polymerase iota (Polι) belongs to the Y-family of DNA polymerases that are involved in DNA damage tolerance through their role in translesion DNA synthesis. Like all other Y-family polymerases, Polι interacts with proliferating cell nuclear antigen (PCNA), Rev1, ubiquitin and ubiquitinated-PCNA and is also ubiquitinated itself. Here, we report that Polι also interacts with the p300 acetyltransferase and is acetylated. The primary acetylation site is K550, located in the Rev1-interacting region. However, K550 amino acid substitutions have no effect on Polι's ability to interact with Rev1. Interestingly, we find that acetylation of Polι significantly and specifically increases in response to SN2 alkylating agents and to a lower extent to SN1 alkylating and oxidative agents. As we have not observed acetylation of Polι's closest paralogue, DNA polymerase eta (Polη), with which Polι shares many functional similarities, we believe that this modification might exclusively regulate yet to be determined, and separate function(s) of Polι.

Publication types

  • Research Support, N.I.H., Intramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylation
  • Alkylating Agents / pharmacology*
  • Amino Acid Motifs
  • Binding Sites
  • DNA Polymerase iota
  • DNA-Directed DNA Polymerase / chemistry
  • DNA-Directed DNA Polymerase / metabolism*
  • HEK293 Cells
  • Humans
  • Nucleotidyltransferases / metabolism
  • Protein Binding
  • Protein Processing, Post-Translational / drug effects
  • p300-CBP Transcription Factors / metabolism

Substances

  • Alkylating Agents
  • p300-CBP Transcription Factors
  • p300-CBP-associated factor
  • Nucleotidyltransferases
  • REV1 protein, human
  • DNA-Directed DNA Polymerase
  • DNA Polymerase iota
  • POLI protein, human