Role of NS5A-L31/Y93 Double Wild-type in Failure of Glecaprevir/Pibrentasvir Double Therapy in Two Patients with a History of Direct-acting Antiviral Agent Failure: An Ultra-deep Sequencing Analysis

Intern Med. 2019 Sep 15;58(18):2657-2662. doi: 10.2169/internalmedicine.2604-18. Epub 2019 Jun 7.

Abstract

We experienced two cases of hepatitis C virus (HCV) eradication failure in patients with a history of non-responsiveness to previous treatments with direct-acting antiviral agents (DAAs) who were subsequently treated with the combination of glecaprevir and pibrentasvir (GLE/PIB). Direct sequencing at commencement of GLE/PIB therapy showed non-structural protein (NS) 5A-P32 deletion in the first patient and NS5A-R30E/Q54H/A92K in the second patient (both genotype 1b). The common point was that L31/Y93 was double wild-type, and the IL28B polymorphism was non-TT type. Even when L31/Y93 is double wild-type, other NS5A mutations may affect the DAA re-treatment outcome. We analyzed the transition of amino acid mutations at NS5A by ultra-deep sequencing.

Keywords: direct-acting antivirals; glecaprevir; hepatitis C virus; pibrentasvir; resistance-associated variants; ultra-deep sequencing.

Publication types

  • Case Reports

MeSH terms

  • Adult
  • Aminoisobutyric Acids
  • Antiviral Agents / therapeutic use*
  • Benzimidazoles / therapeutic use*
  • Cyclopropanes
  • Female
  • Genotype
  • Hepatitis C, Chronic* / drug therapy
  • Hepatitis C, Chronic* / genetics
  • Humans
  • Interferons / genetics*
  • Lactams, Macrocyclic
  • Leucine / analogs & derivatives
  • Polymorphism, Genetic
  • Proline / analogs & derivatives
  • Pyrrolidines
  • Quinoxalines / therapeutic use*
  • Sulfonamides / therapeutic use*

Substances

  • Aminoisobutyric Acids
  • Antiviral Agents
  • Benzimidazoles
  • Cyclopropanes
  • interferon-lambda, human
  • Lactams, Macrocyclic
  • Pyrrolidines
  • Quinoxalines
  • Sulfonamides
  • pibrentasvir
  • Interferons
  • Proline
  • Leucine
  • glecaprevir