Histone demethylase KDM7A is required for stem cell maintenance and apoptosis inhibition in breast cancer

J Cell Physiol. 2020 Feb;235(2):932-943. doi: 10.1002/jcp.29008. Epub 2019 Jun 24.

Abstract

Histone demethylase KDM7A regulates neuronal differentiation and development in mammals. In this study, we found that KDM7A was also required for breast cancer stem cells (BCSCs) maintenance. Silencing KDM7A significantly reduced the BCSCs population and mamosphere formation in vitro, and inhibited breast tumor growth in vivo. Restoring KDM7A expression rescued the defect in stem cell maintenance. Our mechanism analysis suggested that KDM7A upregulated the stemness-associated factors KLF4 and c-MYC for BCSCs maintenance. In addition, KDM7A knockdown promoted apoptosis through decreasing BCL2 expression and BAD phosphorylation in breast cancer (BrCa). Furthermore, restoring KDM7A and BCL2 expression rescued apoptosis inhibition in breast cancer, suggesting that KDM7A inhibited apoptosis by upregulating the BCL2 level in breast cancer. In conclusion, KDM7A promotes cancer stem cell maintenance and apoptosis inhibition in breast cancer.

Keywords: KDM7A; apoptosis; breast cancer stem cell; stem cell maintenance.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenocarcinoma / pathology
  • Animals
  • Apoptosis / genetics*
  • Breast Neoplasms / genetics
  • Breast Neoplasms / pathology*
  • Cell Proliferation / genetics
  • Female
  • Humans
  • Jumonji Domain-Containing Histone Demethylases / genetics*
  • Jumonji Domain-Containing Histone Demethylases / metabolism*
  • Kruppel-Like Factor 4
  • Mice
  • Mice, Nude
  • Neoplastic Stem Cells / pathology*
  • Proto-Oncogene Proteins c-bcl-2 / metabolism
  • RNA Interference
  • RNA, Small Interfering / genetics
  • Spheroids, Cellular
  • Tumor Cells, Cultured
  • Xenograft Model Antitumor Assays
  • bcl-Associated Death Protein / metabolism

Substances

  • BAD protein, human
  • BCL2 protein, human
  • KLF4 protein, human
  • Klf4 protein, mouse
  • Kruppel-Like Factor 4
  • Proto-Oncogene Proteins c-bcl-2
  • RNA, Small Interfering
  • bcl-Associated Death Protein
  • Jumonji Domain-Containing Histone Demethylases
  • KDM7A protein, human