Diverse Structural Conversion and Aggregation Pathways of Alzheimer's Amyloid-β (1-40)

ACS Nano. 2019 Aug 27;13(8):8766-8783. doi: 10.1021/acsnano.9b01578. Epub 2019 Jul 24.

Abstract

Complex amyloid aggregation of amyloid-β (1-40) (Aβ1-40) in terms of monomer structures has not been fully understood. Herein, we report the microscopic mechanism and pathways of Aβ1-40 aggregation with macroscopic viewpoints through tuning its initial structure and solubility. Partial helical structures of Aβ1-40 induced by low solvent polarity accelerated cytotoxic Aβ1-40 amyloid fibrillation, while predominantly helical folds did not aggregate. Changes in the solvent polarity caused a rapid formation of β-structure-rich protofibrils or oligomers via aggregation-prone helical structures. Modulation of the pH and salt concentration transformed oligomers to protofibrils, which proceeded to amyloid formation. We reveal diverse molecular mechanisms underlying Aβ1-40 aggregation with conceptual energy diagrams and propose that aggregation-prone partial helical structures are key to inducing amyloidogenesis. We demonstrate that context-dependent protein aggregation is comprehensively understood using the macroscopic phase diagram, which provides general insights into differentiation of amyloid formation and phase separation from unfolded and folded structures.

Keywords: Alzheimerʼs disease; aggregation pathway; amyloid fibril; amyloid β; helical structure; phase diagram; protein misfolding and aggregation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alzheimer Disease / genetics*
  • Alzheimer Disease / pathology
  • Amyloid / chemistry
  • Amyloid / genetics
  • Amyloid beta-Peptides / chemistry
  • Amyloid beta-Peptides / ultrastructure*
  • Humans
  • Peptide Fragments / chemistry
  • Peptide Fragments / ultrastructure*
  • Protein Aggregation, Pathological / genetics*
  • Protein Conformation, alpha-Helical / genetics*
  • Protein Conformation, beta-Strand / genetics
  • Protein Folding / drug effects
  • Protein Stability / drug effects
  • Signal Transduction / drug effects
  • Solubility

Substances

  • Amyloid
  • Amyloid beta-Peptides
  • Peptide Fragments
  • amyloid beta-protein (1-40)