Synthesis of a trisaccharide of 3-deoxy-D-manno-2-octulopyranosylonic acid (KDO) residues related to the genus-specific lipopolysaccharide epitope of Chlamydia

Carbohydr Res. 1988 Dec 1;183(2):183-99. doi: 10.1016/0008-6215(88)84073-4.

Abstract

The disaccharides, O-(sodium 3-deoxy-alpha- and -beta-D-manno-2-octulopyranosylonate)-(2----8)-sodium (allyl 3-deoxy-alpha-D-manno-2-octulopyranosid)onate, were prepared via glycosylation of methyl (allyl 4,5,7-tri-O-acetyl-3-deoxy-alpha-D-manno-2-octulopyranosid)onat e with methyl (4,5,7,8-tetra-O-acetyl-3-deoxy-D-manno-2-octulopyranosyl bromide)onate under Helferich and Koenigs-Knorr conditions, respectively. Based on g.l.c.-m.s. data of the alpha- and beta-(2----8)-linked disaccharide derivatives, obtained after carbonyl- and carboxyl-group reduction, followed by methylation, the alpha-anomeric configuration was assigned to the terminal KDO-residue in the KDO-region of Chlamydial lipopolysaccharide. The trisaccharide O-(sodium 3-deoxy-alpha-D-manno-2-octulopyranosylonate)-(2----8)-(sodium 3-deoxy-alpha-D-manno-2-octulopyranosylonate)-(2----4)-sodium (allyl 3-deoxy-alpha-D-manno-2-octulopyranosid)onate was obtained via block synthesis using an alpha-(2----8)-linked disaccharide bromide derivative as the glycosyl donor. Copolymerization of the allyl glycosides with acrylamide gave water-soluble macromolecular antigens, suitable for defining epitope specificities of monoclonal antibodies directed against Chlamydial LPS.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acrylamide
  • Acrylamides
  • Antigens, Bacterial*
  • Carbohydrate Conformation
  • Carbohydrate Sequence
  • Chemical Phenomena
  • Chemistry
  • Chlamydia / immunology*
  • Chromatography, Gas
  • Disaccharides / chemical synthesis
  • Gas Chromatography-Mass Spectrometry
  • Glycosylation
  • Lipopolysaccharides*
  • Magnetic Resonance Spectroscopy
  • Methylation
  • Molecular Sequence Data
  • Molecular Structure
  • Polymers
  • Sugar Acids*
  • Trisaccharides* / chemical synthesis*

Substances

  • Acrylamides
  • Antigens, Bacterial
  • Disaccharides
  • Lipopolysaccharides
  • Polymers
  • Sugar Acids
  • Trisaccharides
  • 2-keto-3-deoxyoctonate
  • Acrylamide