A Case Report: Rapid Micro-Induction of Buprenorphine/Naloxone to Administer Buprenorphine Extended-Release in an Adolescent With Severe Opioid Use Disorder

Am J Addict. 2020 Nov;29(6):531-535. doi: 10.1111/ajad.13050. Epub 2020 Apr 29.

Abstract

Background and objectives: Buprenorphine extended-release (BUP-XR) is a monthly injectable form of opioid agonist therapy. Before its administration, a minimum 7-day induction period with a transmucosal buprenorphine-containing product is recommended.

Methods: Case report (n = 1).

Results: A 16-year-old female with active, severe opioid use disorder (OUD) and stimulant use disorder, hepatitis C virus, co-occurring mental health disorders, and complex social stressors had five recent overdoses requiring naloxone. She had previously been treated with methadone and several trials of sublingual buprenorphine/naloxone, but would quickly discontinue the treatment. Using a rapid micro-induction protocol, buprenorphine/naloxone was administered for 3 days. On day 4, 300 mg BUP-XR was administered subcutaneously. Minimal withdrawal symptoms occurred, despite recent fentanyl use.

Discussion and conclusions: A rapid sublingual buprenorphine/naloxone micro-induction was successfully used to initiate BUP-XR, thereby eliminating the abstinence period prior to buprenorphine/naloxone administration, shortening the induction period, and minimizing withdrawal.

Scientific significance: This is the first reported case of using rapid micro-induction as a bridge to initiate BUP-XR. By reducing the length of induction to 4 days and minimizing withdrawal, this induction method can make BUP-XR more accessible to patients who would otherwise refuse the medication due to concerns of enduring withdrawal. (Am J Addict 2020;29:531-535).

Publication types

  • Case Reports
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Sublingual
  • Adolescent
  • Buprenorphine / administration & dosage
  • Buprenorphine / therapeutic use
  • Buprenorphine, Naloxone Drug Combination / administration & dosage*
  • Buprenorphine, Naloxone Drug Combination / therapeutic use
  • Delayed-Action Preparations / administration & dosage
  • Delayed-Action Preparations / therapeutic use
  • Drug Administration Schedule
  • Female
  • Humans
  • Induction Chemotherapy / methods*
  • Narcotic Antagonists / administration & dosage*
  • Narcotic Antagonists / therapeutic use
  • Opioid-Related Disorders / drug therapy*

Substances

  • Buprenorphine, Naloxone Drug Combination
  • Delayed-Action Preparations
  • Narcotic Antagonists
  • Buprenorphine