Differential detection of M184V/I between plasma historical HIV genotypes and HIV proviral DNA from PBMCs

J Antimicrob Chemother. 2020 Aug 1;75(8):2249-2252. doi: 10.1093/jac/dkaa146.

Abstract

Background: The M184V/I reverse transcriptase mutation, which confers major resistance to lamivudine and emtricitabine, is still quite frequent in people living with HIV. The underlying presence of the M184V/I mutation may undermine virological outcomes of ART, particularly in the context of proposed treatment with two-drug combinations that include drugs affected by M184V, such as lamivudine. In suppressed patients for whom historical data are seldom available, resistance assays evaluating integrated viral DNA can help select a fully active switch regimen.

Objectives: To compare detectability of M184V/I in historical HIV-1 RNA analyses versus HIV-1 DNA sequencing.

Methods: We analysed the detection of the M184V/I mutation in a prospective study and compared HIV historical genotypes (plasma) versus integrated HIV DNA (PBMCs) obtained via a validated commercial proviral HIV DNA assay. Eligible participants had HIV-1 RNA <50 copies/mL for ≥6 consecutive months prior to screening. A plasma historical genotypic report (HGR) showing the presence of M184V/I was required for all participants and proviral HIV DNA analysis was conducted prior to enrolment.

Results: All 84 participants had evidence of M184V or M184I in their HGR (100%), whereas the mutation was detected in only 40/84 participants by proviral HIV DNA sequencing analysis (48%). Differential detection of M184V/I was not associated with timing differences between the HGR and proviral HIV DNA sampling, the overall duration of ART, or CD4 cell counts and HIV-1 viral load at baseline.

Conclusions: Our results suggest that undetected M184V/I should be considered when switching virologically suppressed patients to new regimens, particularly two-drug lamivudine- or emtricitabine-containing combinations.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Anti-HIV Agents* / pharmacology
  • Anti-HIV Agents* / therapeutic use
  • Drug Resistance, Viral
  • Genotype
  • HIV Infections* / drug therapy
  • HIV-1* / genetics
  • Humans
  • Lamivudine / therapeutic use
  • Mutation
  • Pharmaceutical Preparations*
  • Prospective Studies
  • Viral Load

Substances

  • Anti-HIV Agents
  • Pharmaceutical Preparations
  • Lamivudine