Mutations in PIGA cause a CD52-/GPI-anchor-deficient phenotype complicating alemtuzumab treatment in T-cell prolymphocytic leukemia

Eur J Haematol. 2020 Dec;105(6):786-796. doi: 10.1111/ejh.13511. Epub 2020 Sep 28.

Abstract

Objective: Infusional alemtuzumab followed by consolidating allogeneic hematopoietic stem cell transplantation in eligible patients is considered a standard of care in T-cell prolymphocytic leukemia (T-PLL). Antibody selection against CD52 has been associated with the development of CD52-negative leukemic T cells at time of relapse. Clinical implications and molecular mechanisms underlying this phenotypic switch are unknown.

Methods: We performed flow cytometry and real-time-PCR for CD52-expression and next generation sequencing for PIGA mutational analyses.

Results: We identified loss of CD52 expression after alemtuzumab treatment in two of 21 T-PLL patients resulting from loss of GPI-anchor expression caused by inactivating mutations of the PIGA gene. One patient with relapsed T-PLL exhibited a single PIGA mutation, causing a CD52-negative escape variant of the initial leukemic cell clone, preventing alemtuzumab-retreatment. The second patient with continued complete remission after alemtuzumab treatment harbored three different PIGA mutations that affected either the non-neoplastic T cell or the mononuclear cell compartment and resulted in symptomatic paroxysmal nocturnal hemoglobinuria. Next generation sequencing of T-PLL cells collected before the initiation of treatment revealed PIGA wild-type sequence reads in all 16 patients with samples available for testing.

Conclusion: These data indicate that PIGA mutations were acquired during or after completion of alemtuzumab treatment.

Keywords: CD52; PIGA; PNH; T-PLL; T-cell prolymphocytic leukemia; alemtuzumab.

MeSH terms

  • Alemtuzumab / pharmacology*
  • Alemtuzumab / therapeutic use
  • CD52 Antigen / genetics*
  • CD52 Antigen / metabolism
  • DNA Mutational Analysis
  • Gene Expression Regulation, Leukemic / drug effects
  • High-Throughput Nucleotide Sequencing
  • Humans
  • Immunophenotyping
  • Leukemia, Prolymphocytic, T-Cell / drug therapy
  • Leukemia, Prolymphocytic, T-Cell / genetics*
  • Leukemia, Prolymphocytic, T-Cell / metabolism
  • Membrane Proteins / genetics*
  • Membrane Proteins / metabolism
  • Mutation*
  • Phenotype
  • T-Lymphocytes / drug effects*
  • T-Lymphocytes / metabolism*
  • T-Lymphocytes / pathology

Substances

  • CD52 Antigen
  • CD52 protein, human
  • Membrane Proteins
  • phosphatidylinositol glycan-class A protein
  • Alemtuzumab