BDNF rs6265 Variant Alters Outcomes with Levodopa in Early-Stage Parkinson's Disease

Neurotherapeutics. 2020 Oct;17(4):1785-1795. doi: 10.1007/s13311-020-00965-9. Epub 2020 Nov 19.

Abstract

Disease outcomes are heterogeneous in Parkinson's disease and may be predicted by gene variants. This study investigated if the BDNF rs6265 single nucleotide polymorphism (SNP) is associated with differential outcomes with specific pharmacotherapy treatment strategies in the "NIH Exploratory Trials in PD Long-term Study 1" (NET-PD LS-1, n = 540). DNA samples were genotyped for the rs6265 SNP and others (rs11030094, rs10501087, rs1491850, rs908867, and rs1157659). The primary measures were the Unified Parkinson's Disease Rating Scale (UPDRS) and its motor component (UPDRS-III). Groups were divided by genotype and treatment regimen (levodopa monotherapy vs levodopa with other medications vs no levodopa). T allele carriers were associated with worse UPDRS outcomes compared to C/C subjects when treated with levodopa monotherapy (+ 6 points, p = 0.02) and to T allele carriers treated with no levodopa treatment strategies (UPDRS: + 8 points, p = 0.01; UPDRS-III: + 6 points, p = 0.01). Similar effects of worse outcomes associated with levodopa monotherapy were observed in the BDNF rs11030094, rs10501087, and rs1491850 SNPs. This study suggests the levodopa monotherapy strategy is associated with worse disease outcomes in BDNF rs6265 T carriers. Pending prospective validation, BDNF variants may be precision medicine factors to consider for symptomatic treatment decisions for early-stage PD patients.

Keywords: Brain-derived neurotrophic factor; Levodopa; Parkinson disease; Subthalamic nucleus deep brain stimulation; rs6265.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antiparkinson Agents / therapeutic use*
  • Brain-Derived Neurotrophic Factor / genetics*
  • Early Diagnosis
  • Female
  • Genetic Variation / genetics*
  • Humans
  • Levodopa / therapeutic use*
  • Longitudinal Studies
  • Male
  • Parkinson Disease / diagnosis
  • Parkinson Disease / drug therapy*
  • Parkinson Disease / genetics*
  • Retrospective Studies
  • Treatment Outcome

Substances

  • Antiparkinson Agents
  • Brain-Derived Neurotrophic Factor
  • Levodopa
  • BDNF protein, human