Selective cine-arylation of tert-cyclobutanols with indoles enabled by nickel catalysis

Chem Commun (Camb). 2021 May 11;57(38):4686-4689. doi: 10.1039/d1cc01233a.

Abstract

In previous literature, tert-cyclobutanols are widely studied for C-C bond activation exclusively leading to the formation of ordinary γ-substituted ketones. Herein, we first report a nickel-catalyzed cine-arylation of tert-cyclobutanols with indoles to access β-aryl ketones with an unusual site-selectivity at the C3-position of tert-cyclobutanols. The reaction features earth-abundant nickel catalysis, excellent regioselectivity, high atom-economy, and broad substrate scope.