ERG transcription factors have a splicing regulatory function involving RBFOX2 that is altered in the EWS-FLI1 oncogenic fusion

Nucleic Acids Res. 2021 May 21;49(9):5038-5056. doi: 10.1093/nar/gkab305.

Abstract

ERG family proteins (ERG, FLI1 and FEV) are a subfamily of ETS transcription factors with key roles in physiology and development. In Ewing sarcoma, the oncogenic fusion protein EWS-FLI1 regulates both transcription and alternative splicing of pre-messenger RNAs. However, whether wild-type ERG family proteins might regulate splicing is unknown. Here, we show that wild-type ERG proteins associate with spliceosomal components, are found on nascent RNAs, and induce alternative splicing when recruited onto a reporter minigene. Transcriptomic analysis revealed that ERG and FLI1 regulate large numbers of alternative spliced exons (ASEs) enriched with RBFOX2 motifs and co-regulated by this splicing factor. ERG and FLI1 are associated with RBFOX2 via their conserved carboxy-terminal domain, which is present in EWS-FLI1. Accordingly, EWS-FLI1 is also associated with RBFOX2 and regulates ASEs enriched in RBFOX2 motifs. However, in contrast to wild-type ERG and FLI1, EWS-FLI1 often antagonizes RBFOX2 effects on exon inclusion. In particular, EWS-FLI1 reduces RBFOX2 binding to the ADD3 pre-mRNA, thus increasing its long isoform, which represses the mesenchymal phenotype of Ewing sarcoma cells. Our findings reveal a RBFOX2-mediated splicing regulatory function of wild-type ERG family proteins, that is altered in EWS-FLI1 and contributes to the Ewing sarcoma cell phenotype.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alternative Splicing*
  • Calmodulin-Binding Proteins / genetics
  • Calmodulin-Binding Proteins / metabolism
  • Cell Line
  • Cell Line, Tumor
  • HeLa Cells
  • Human Umbilical Vein Endothelial Cells / metabolism
  • Humans
  • Oncogene Proteins, Fusion / metabolism*
  • Protein Domains
  • Proto-Oncogene Protein c-fli-1 / metabolism*
  • RNA Splicing Factors / metabolism*
  • RNA-Binding Protein EWS / metabolism*
  • Repressor Proteins / metabolism*
  • Sarcoma, Ewing / genetics
  • Sarcoma, Ewing / metabolism
  • Transcriptional Regulator ERG / chemistry
  • Transcriptional Regulator ERG / metabolism

Substances

  • ADD3 protein, human
  • Calmodulin-Binding Proteins
  • ERG protein, human
  • EWS-FLI fusion protein
  • FLI1 protein, human
  • Oncogene Proteins, Fusion
  • Proto-Oncogene Protein c-fli-1
  • RBFOX2 protein, human
  • RNA Splicing Factors
  • RNA-Binding Protein EWS
  • Repressor Proteins
  • Transcriptional Regulator ERG