Identification and evaluation of antiviral potential of thymoquinone, a natural compound targeting Chikungunya virus capsid protein

Virology. 2021 Sep:561:36-46. doi: 10.1016/j.virol.2021.05.013. Epub 2021 Jun 10.

Abstract

Capsid protein (CP) of Chikungunya virus (CHIKV) is a multifunctional protein with a conserved hydrophobic pocket that plays a crucial role in the capsid assembly and virus budding process. This study demonstrates antiviral activity of thymoquinone (TQ), a natural compound targeting the hydrophobic pocket of CP. The binding of TQ to the hydrophobic pocket of CHIKV CP was analysed by structure-based molecular docking, isothermal titration calorimetry and fluorescence spectroscopy. The binding constant KD obtained for TQ was 27 μM. Additionally, cell-based antiviral studies showed that TQ diminished CHIKV replication with an EC50 value 4.478 μM. Reduction in viral RNA copy number and viral replication as assessed by the qRT-PCR and immunofluorescence assay, confirmed the antiviral potential of TQ. Our study reveals that TQ is an effective antiviral targeting the hydrophobic pocket of CHIKV CP and may serve as the basis for development of a broad-spectrum therapy against alphaviral diseases.

Keywords: Antiviral activity; Capsid protein; Chikungunya virus; Hydrophobic pocket; Natural compound; Thymoquinone.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antiviral Agents / metabolism
  • Antiviral Agents / pharmacology*
  • Benzoquinones / metabolism
  • Benzoquinones / pharmacology*
  • Capsid Proteins / chemistry
  • Capsid Proteins / metabolism*
  • Cell Survival / drug effects
  • Chikungunya virus / drug effects*
  • Chikungunya virus / physiology
  • Chlorocebus aethiops
  • Hydrophobic and Hydrophilic Interactions
  • Microbial Sensitivity Tests
  • Models, Molecular
  • Molecular Docking Simulation
  • Protein Binding
  • Protein Conformation
  • Vero Cells
  • Virus Replication / drug effects

Substances

  • Antiviral Agents
  • Benzoquinones
  • Capsid Proteins
  • thymoquinone