Unravelling the antifungal mode of action of curcumin by potential inhibition of CYP51B: A computational study validated in vitro on mucormycosis agent, Rhizopus oryzae

Arch Biochem Biophys. 2021 Nov 15:712:109048. doi: 10.1016/j.abb.2021.109048. Epub 2021 Sep 30.

Abstract

Like human, fungi too are known to share lot of structural similarities amongst their CYPs (Cytochrome P450 super family of enzymes) which allows antifungal 'azole' compounds to interact with CYPs of human. Clotrimazole, an 'azole' antifungal drug, is a known inhibitor of fungal CYP named CYP51B. Curcumin, a phytochemical obtained from Curcuma longa has the ability to interact with several different human CYPs to induce inhibition. The sequence and the structural similarities amongst both human and fungal CYPs suggest a strong possibility for curcumin to interact with fungal CYP51B to behave like an antifungal agent. To test this hypothesis a study was designed involving mucormycosis agent, Rhizopus oryzae. The ability of curcumin to interact with fungal CYP51B was analysed computationally through molecular docking, MM-GBSA and Molecular Dynamics (MD) simulation assessment. Further, interaction profile for fungal CYP51B-curcumin was compared with human CYP3A4-curcumin, as there are published evidence describing curcumin as an inhibitor of human CYPs. Additionally, to validate in silico findings, an in vitro assay was performed to examine the antifungal potentials of curcumin on the R. oryzae. Conclusive results allow us to determine a plausible mode of action of curcumin to act as an antifungal against a mucormycosis agent.

Keywords: Antifungal; CYP51B; Curcumin; Cytochrome P450; Mucormycosis; Rhizopus oryzae.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Antifungal Agents / metabolism
  • Antifungal Agents / pharmacology*
  • Clotrimazole / metabolism
  • Clotrimazole / pharmacology
  • Curcumin / metabolism
  • Curcumin / pharmacology*
  • Cytochrome P-450 Enzyme Inhibitors / metabolism
  • Cytochrome P-450 Enzyme Inhibitors / pharmacology*
  • Cytochrome P-450 Enzyme System / metabolism*
  • Ergosterol / metabolism
  • Fungal Proteins / antagonists & inhibitors*
  • Fungal Proteins / metabolism
  • Humans
  • Microbial Sensitivity Tests
  • Molecular Docking Simulation
  • Molecular Dynamics Simulation
  • Phylogeny
  • Protein Binding
  • Rhizopus oryzae / drug effects*

Substances

  • Antifungal Agents
  • Cytochrome P-450 Enzyme Inhibitors
  • Fungal Proteins
  • Cytochrome P-450 Enzyme System
  • Clotrimazole
  • Curcumin
  • Ergosterol