Factors affecting the rheological behaviour of carbomer dispersions in hydroalcoholic medium: Towards the optimization of hand sanitiser gel formulations

Int J Pharm. 2022 Mar 25:616:121503. doi: 10.1016/j.ijpharm.2022.121503. Epub 2022 Jan 24.

Abstract

Hand sanitizers represent a primary measure for the prevention of transmissible infections, whose use has been greatly increased during CoViD-19 pandemic. Most of the commercially available products are hydrogels, employing carbomers as thickening agents. However, few information is still available regarding performances of carbomers in hydroalcoholic media containing a percentage of alcohols ≥ 60% v/v as recommended for disinfection. The aim of this study was to investigate the colloidal behaviour of carbomer 974 and carbomer 980 in hydroalcoholic media containing from 50 to 80% w/w of alcohol (ethanol or isopropanol) and neutralised with triethanolamine or aminomethyl propanol. Both carbomers provide transparent hydrogels in water, but carbomer 980 should be preferred for the formulation of hydrogel with a percentage of alcohol ≥ 50% w/w for its better solvation. The critical alcohol concentration (CAlC), above which polymer precipitation occurs, depends on the type of alcohol and base used. Carbomer dispersions with a higher content of alcohol can be prepared using aminomethyl propanol rather than triethanolamine. The choice of the more suitable components is fundamental for the isopropanol-based dispersions since the CAlC is closer to the recommended concentrations for disinfection. Overall, these results provide helpful insights for the correct preparation of alcohol-based hand sanitizers using carbomers.

Keywords: Carbopol; Hydrogels; Rheology; Transmittance; Viscosity; pH.

MeSH terms

  • Acrylic Resins
  • COVID-19*
  • Ethanol
  • Hand Sanitizers*
  • Humans
  • Pandemics
  • Rheology
  • SARS-CoV-2
  • Viscosity

Substances

  • Acrylic Resins
  • Hand Sanitizers
  • carbomer
  • Ethanol