Chronic Systemic Dexamethasone Regulates the Mineralocorticoid/Glucocorticoid Pathways Balance in Rat Ocular Tissues

Int J Mol Sci. 2022 Jan 24;23(3):1278. doi: 10.3390/ijms23031278.

Abstract

Central serous chorioretinopathy (CSCR) is a retinal disease affecting the retinal pigment epithelium (RPE) and the choroid. This is a recognized side-effect of glucocorticoids (GCs), administered through nasal, articular, oral and dermal routes. However, CSCR does not occur after intraocular GCs administration, suggesting that a hypothalamic-pituitary-adrenal axis (HPA) brake could play a role in the mechanistic link between CSCR and GS. The aim of this study was to explore this hypothesis. To induce HPA brake, Lewis rats received a systemic injection of dexamethasone daily for five days. Control rats received saline injections. Baseline levels of corticosterone were measured by Elisa at baseline and at 5 days in the serum and the ocular media and dexamethasone levels were measured at 5 days in the serum and ocular media. The expression of genes encoding glucocorticoid receptor (GR), mineralocorticoid receptors (MR), and the 11 beta hydroxysteroid dehydrogenase (HSD) enzymes 1 and 2 were quantified in the neural retina and in RPE/ choroid. The expression of MR target genes was quantified in the retina (Scnn1A (encoding ENac-α, Kir4.1 and Aqp4) and in the RPE/choroid (Shroom 2, Ngal, Mmp9 and Omg, Ptx3, Plaur and Fosl-1). Only 10% of the corticosterone serum concentration was measured in the ocular media. Corticosterone levels in the serum and in the ocular media dropped after 5 days of dexamethasone systemic treatment, reflecting HPA axis brake. Whilst both GR and MR were downregulated in the retina without MR/GR imbalance, in the RPE/choroid, both MR/GR and 11β-hsd2/11β-hsd1 ratio increased, indicating MR pathway activation. MR-target genes were upregulated in the RPE/ choroid but not in the retina. The psychological stress induced by the repeated injection of saline also induced HPA axis brake with a trend towards MR pathway activation in RPE/ choroid. HPA axis brake causes an imbalance of corticoid receptors expression in the RPE/choroid towards overactivation of MR pathway, which could favor the occurrence of CSCR.

Keywords: central serous chorioretinopathy; glucocorticoid; mineralocorticoid; retina.

MeSH terms

  • Animals
  • Central Serous Chorioretinopathy / drug therapy
  • Central Serous Chorioretinopathy / physiopathology
  • Choroid / drug effects
  • Choroid / metabolism
  • Corticosterone / blood
  • Dexamethasone / metabolism
  • Dexamethasone / pharmacology
  • Eye / metabolism
  • Glucocorticoids / metabolism*
  • Hypothalamo-Hypophyseal System / metabolism
  • Mineralocorticoids / metabolism*
  • Ocular Physiological Phenomena / drug effects
  • Pituitary-Adrenal System / metabolism
  • Rats
  • Rats, Inbred Lew
  • Receptors, Glucocorticoid / metabolism
  • Retina / drug effects
  • Retina / metabolism*
  • Retinal Pigment Epithelium / drug effects
  • Retinal Pigment Epithelium / metabolism
  • Signal Transduction / genetics
  • Signal Transduction / physiology

Substances

  • Glucocorticoids
  • Mineralocorticoids
  • Receptors, Glucocorticoid
  • Dexamethasone
  • Corticosterone