HOXD8 hypermethylation as a fully sensitive and specific biomarker for biliary tract cancer detectable in tissue and bile samples

Br J Cancer. 2022 Jun;126(12):1783-1794. doi: 10.1038/s41416-022-01738-1. Epub 2022 Feb 17.

Abstract

Background: Biliary tract cancers (BTC) are rare but highly aggressive tumours with poor prognosis, usually detected at advanced stages. Herein, we aimed at identifying BTC-specific DNA methylation alterations.

Methods: Study design included statistical power and sample size estimation. A genome-wide methylation study of an explorative cohort (50 BTC and ten matched non-tumoral tissue samples) has been performed. BTC-specific altered CpG islands were validated in over 180 samples (174 BTCs and 13 non-tumoral controls). The final biomarkers, selected by a machine-learning approach, were validated in independent tissue (18 BTCs, 14 matched non-tumoral samples) and bile (24 BTCs, five non-tumoral samples) replication series, using droplet digital PCR.

Results: We identified and successfully validated BTC-specific DNA methylation alterations in over 200 BTC samples. The two-biomarker panel, selected by an in-house algorithm, showed an AUC > 0.97. The best-performing biomarker (chr2:176993479-176995557), associated with HOXD8, a pivotal gene in cancer-related pathways, achieved 100% sensitivity and specificity in a new series of tissue and bile samples.

Conclusions: We identified a novel fully efficient BTC biomarker, associated with HOXD8 gene, detectable both in tissue and bile by a standardised assay ready-to-use in clinical trials also including samples from non-invasive matrices.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Bile
  • Biliary Tract Neoplasms* / genetics
  • Biliary Tract Neoplasms* / pathology
  • Biomarkers, Tumor / genetics
  • DNA Methylation*
  • Homeodomain Proteins* / genetics
  • Humans
  • Mutation
  • Transcription Factors* / genetics

Substances

  • Biomarkers, Tumor
  • Homeodomain Proteins
  • Transcription Factors
  • HOXD8 protein, human