β-Catenin-Specific Inhibitor, iCRT14, Promotes BoHV-1 Infection-Induced DNA Damage in Human A549 Lung Adenocarcinoma Cells by Enhancing Viral Protein Expression

Int J Mol Sci. 2022 Feb 19;23(4):2328. doi: 10.3390/ijms23042328.

Abstract

Oncolytic bovine herpesvirus type 1 (BoHV-1) infection induces DNA damage in human lung adenocarcinoma cell line A549. However, the underlying mechanisms are not fully understood. We found that BoHV-1 infection decreased the steady-state protein levels of p53-binding protein 1 (53BP1), which plays a central role in dictating DNA damage repair and maintaining genomic stability. Furthermore, BoHV-1 impaired the formation of 53BP1 foci, suggesting that BoHV-1 inhibits 53BP1-mediated DNA damage repair. Interestingly, BoHV-1 infection redistributed intracellular β-catenin, and iCRT14 (5-[[2,5-Dimethyl-1-(3-pyridinyl)-1H-pyrrol-3-yl]methylene]-3-phenyl-2,4-thiazolidinedione), a β-catenin-specific inhibitor, enhanced certain viral protein expression, such as the envelope glycoproteins gC and gD, and enhanced virus infection-induced DNA damage. Therefore, for the first time, we provide evidence showing that BoHV-1 infection disrupts 53BP1-mediated DNA damage repair and suggest β-catenin as a potential host factor restricting both virus replication and DNA damage in A549 cells.

Keywords: 53BP1; BoHV-1; DNA damage; β-catenin; γH2AX.

MeSH terms

  • A549 Cells
  • Adenocarcinoma of Lung / genetics*
  • Cell Line, Tumor
  • DNA Damage / drug effects*
  • DNA Damage / genetics
  • Herpesviridae Infections / genetics*
  • Herpesvirus 1, Bovine / pathogenicity
  • Humans
  • Lung Neoplasms / genetics*
  • Pyridines / pharmacology*
  • Pyrroles / pharmacology*
  • Thiazolidinediones / pharmacology*
  • Viral Proteins / genetics*
  • Virus Replication / drug effects
  • beta Catenin / antagonists & inhibitors*

Substances

  • Pyridines
  • Pyrroles
  • Thiazolidinediones
  • Viral Proteins
  • beta Catenin
  • iCRT14