Pentoxifylline as an adjunctive in treatment of negative symptoms in chronic schizophrenia: A double-blind, randomized, placebo-controlled trial

CNS Neurosci Ther. 2023 Jan;29(1):354-364. doi: 10.1111/cns.14010. Epub 2022 Nov 7.

Abstract

Aim: The aim of this study was to explore the effectiveness and safety of pentoxifylline as an adjuvant to risperidone in mitigating the negative symptoms in patients with chronic schizophrenia.

Methods: In this randomized, placebo-controlled study, eighty outpatients with chronic schizophrenia were given risperidone for 8 weeks along with either pentoxifylline or a placebo. The positive and negative syndrome scale (PANSS) was used to assess patients at the start of the trial, as well as at 2, 4, 6, and 8 weeks. Pre- and posttreatment serum levels of cAMP, TNF-α-, and IL-6 were measured.

Results: The pentoxifylline group revealed a significant effect for time-treatment interaction on PANSS-negative subscale scores (p < 0.001), PANSS general psychopathology subscale scores (p < 0.001), and PANSS total scores (p < 0.001), but not on PANSS-positive subscale scores (p = 0.169). Additionally, when compared to the placebo group, the pentoxifylline group demonstrated a statistically significant increase in cAMP serum level and a statistically significant decrease in TNF-α and IL-6 serum levels.

Conclusion: Pentoxifylline adjunctive therapy with risperidone for 8 weeks was found to be promising in mitigating the negative symptoms in patients with chronic schizophrenia.

Trial registration number: NCT04094207.

Keywords: PANSS; inflammatory cytokines; negative symptoms; pentoxifylline; phosphodiesterase inhibitor; schizophrenia.

Publication types

  • Randomized Controlled Trial
  • Retracted Publication

MeSH terms

  • Antipsychotic Agents* / therapeutic use
  • Double-Blind Method
  • Drug Therapy, Combination
  • Humans
  • Interleukin-6
  • Pentoxifylline* / therapeutic use
  • Psychiatric Status Rating Scales
  • Risperidone / therapeutic use
  • Schizophrenia* / diagnosis
  • Schizophrenia* / drug therapy
  • Schizophrenic Psychology
  • Treatment Outcome
  • Tumor Necrosis Factor-alpha

Substances

  • Risperidone
  • Antipsychotic Agents
  • Pentoxifylline
  • Tumor Necrosis Factor-alpha
  • Interleukin-6

Associated data

  • ClinicalTrials.gov/NCT04094207