[Pharmacokinetic studies of a new oral cephem T-2588. Pharmacokinetics in gastrectomized volunteers and the renal excretory system in healthy volunteers]

Jpn J Antibiot. 1986 Oct;39(10):2701-9.
[Article in Japanese]

Abstract

According to the result of the pharmacokinetic examination of T-2588 (esterified prodrug of T-2525) administered to adult male volunteers who have undergone gastrectomy, it appears that the absorption of T-2588 is delayed in the hypoacidity or the anacidity and also the excretion ratio of T-2525A (an inactive metabolite of T-2525) showed a tendency to become higher in these subjects. Again, according to the result of the pharmacokinetic examination of T-2588 when it was administered together with probenecid to normal healthy volunteers, it appears that the T-2525 is excreted from the kidneys not only into the glomerular filtration but also partly through renal tubules.

Publication types

  • English Abstract

MeSH terms

  • Adult
  • Cefmenoxime* / analogs & derivatives*
  • Cephalosporins / metabolism*
  • Gastrectomy*
  • Glomerular Filtration Rate
  • Humans
  • Kidney / metabolism*
  • Kinetics
  • Male
  • Tissue Distribution

Substances

  • Cephalosporins
  • cefteram pivoxil
  • Cefmenoxime