Isobutyric acid enhances the anti-tumour effect of anti-PD-1 antibody

Sci Rep. 2024 May 17;14(1):11325. doi: 10.1038/s41598-024-59677-1.

Abstract

The low response rate of immune checkpoint inhibitors (ICIs) is a challenge. The efficacy of ICIs is influenced by the tumour microenvironment, which is controlled by the gut microbiota. In particular, intestinal bacteria and their metabolites, such as short chain fatty acids (SCFAs), are important regulators of cancer immunity; however, our knowledge on the effects of individual SCFAs remains limited. Here, we show that isobutyric acid has the strongest effect among SCFAs on both immune activity and tumour growth. In vitro, cancer cell numbers were suppressed by approximately 75% in humans and mice compared with those in controls. Oral administration of isobutyric acid to carcinoma-bearing mice enhanced the effect of anti-PD-1 immunotherapy, reducing tumour volume by approximately 80% and 60% compared with those in the control group and anti-PD-1 antibody alone group, respectively. Taken together, these findings may support the development of novel cancer therapies that can improve the response rate to ICIs.

MeSH terms

  • Animals
  • Cell Line, Tumor
  • Drug Synergism
  • Fatty Acids, Volatile / metabolism
  • Fatty Acids, Volatile / pharmacology
  • Female
  • Gastrointestinal Microbiome / drug effects
  • Humans
  • Immune Checkpoint Inhibitors* / pharmacology
  • Immune Checkpoint Inhibitors* / therapeutic use
  • Immunotherapy / methods
  • Isobutyrates* / pharmacology
  • Mice
  • Neoplasms / drug therapy
  • Neoplasms / immunology
  • Neoplasms / pathology
  • Programmed Cell Death 1 Receptor* / antagonists & inhibitors
  • Tumor Microenvironment* / drug effects
  • Tumor Microenvironment* / immunology

Substances

  • Fatty Acids, Volatile
  • Immune Checkpoint Inhibitors
  • Programmed Cell Death 1 Receptor
  • isobutyric acid
  • Isobutyrates