Nucleoside/nucleotide reverse transcriptase inhibitor-associated weight gain in people living with HIV: data from the Copenhagen Comorbidity in HIV Infection (COCOMO) study

AIDS Care. 2024 Nov;36(11):1635-1646. doi: 10.1080/09540121.2024.2383871. Epub 2024 Aug 20.

Abstract

Weight gain effects of Nucleoside/Nucleotide Reverse Transcriptase Inhibitors in people with HIV (PWH) have been sparsely studied.Participants were enrolled in the Copenhagen Comorbidity in HIV Infection (COCOMO) study. PWH receiving a backbone of emtricitabine, or lamivudine combined with abacavir, tenofovir disoproxil, or tenofovir alafenamide were analysed. Weight gain according to ART backbone and to the third drug was analysed using a multiple linear regression model. Non-ART risk factors were also determined using multiple linear regression.A total of 591 participants were included in the analysis. The majority were middle-aged, virally suppressed males with a mean BMI just above the normal range. Both tenofovir disoproxil/emtricitabine or lamivudine and abacavir /emtricitabine or lamivudine, but not tenofovir alafenamide /emtricitabine or lamivudine were associated with weight gain over two years (0.6 kg, p = 0.025; 1.0 kg, p = 0.005). The third drugs associated with weight increase were non-nucleoside reverse transcriptase inhibitors (NNRTI) (p = 0.035), dolutegravir (p = 0.008) and atazanavir (p = 0.040). Non-ART risk factors for gaining weight were low or normal BMI, age <40 years, underweight, inactivity or highly active at baseline.Tenofovir disoproxil and abacavir-based ART regimens were associated with a small weight gain. Third drug NNRTI, dolutegravir and atazanavir were associated with an increase in weight.

Keywords: ART; HIV; Human immunodeficiency virus; antiretroviral therapy; comorbidity; weight.

MeSH terms

  • Adenine / adverse effects
  • Adenine / analogs & derivatives
  • Adenine / therapeutic use
  • Adult
  • Alanine / therapeutic use
  • Anti-HIV Agents* / adverse effects
  • Anti-HIV Agents* / therapeutic use
  • Comorbidity
  • Cyclopropanes
  • Denmark / epidemiology
  • Dideoxyadenosine / analogs & derivatives
  • Dideoxynucleosides* / adverse effects
  • Dideoxynucleosides* / therapeutic use
  • Emtricitabine / adverse effects
  • Emtricitabine / therapeutic use
  • Female
  • HIV Infections* / drug therapy
  • HIV Infections* / epidemiology
  • Heterocyclic Compounds, 3-Ring / adverse effects
  • Heterocyclic Compounds, 3-Ring / therapeutic use
  • Humans
  • Lamivudine / adverse effects
  • Lamivudine / therapeutic use
  • Male
  • Middle Aged
  • Oxazines
  • Piperazines / adverse effects
  • Pyridones / adverse effects
  • Reverse Transcriptase Inhibitors* / adverse effects
  • Reverse Transcriptase Inhibitors* / therapeutic use
  • Risk Factors
  • Tenofovir* / adverse effects
  • Tenofovir* / analogs & derivatives
  • Tenofovir* / therapeutic use
  • Weight Gain* / drug effects

Substances

  • Reverse Transcriptase Inhibitors
  • Anti-HIV Agents
  • Tenofovir
  • Dideoxynucleosides
  • Emtricitabine
  • abacavir
  • Pyridones
  • Lamivudine
  • Heterocyclic Compounds, 3-Ring
  • Piperazines
  • tenofovir alafenamide
  • dolutegravir
  • Adenine
  • Alanine
  • Cyclopropanes
  • Oxazines
  • Dideoxyadenosine