Effect of alpha-difluoromethylornithine, an irreversible ornithine decarboxylase inhibitor, on formation of GGTase-positive foci

J Toxicol Environ Health. 1983 Apr-Jun;11(4-6):637-41. doi: 10.1080/15287398309530373.

Abstract

The importance of the induction of ornithine decarboxylase to the development of GGTase foci is examined in the classic initiation-promotion assay. This was accomplished by examining the complete foci system in the presence and absence of alpha-DFMO, an irreversible inhibitor of ornithine decarboxylase, at concentrations capable of inhibiting both phenobarbital stimulated and control levels of the enzyme. Although the hepatic enzyme was inhibited by the alpha-DFMO, there was no decrease in the progression of formation of the GGTase foci.

MeSH terms

  • Animals
  • Eflornithine
  • Enzyme Induction / drug effects
  • Liver / enzymology
  • Male
  • Ornithine / analogs & derivatives*
  • Ornithine / pharmacology
  • Ornithine Decarboxylase Inhibitors*
  • Phenobarbital / pharmacology
  • Rats
  • Rats, Inbred F344
  • gamma-Glutamyltransferase / analysis*

Substances

  • Ornithine Decarboxylase Inhibitors
  • Ornithine
  • gamma-Glutamyltransferase
  • Phenobarbital
  • Eflornithine