[Drug sensitivity of Plasmodium falciparum in Madagascar. V. Study of the in vitro activity of quinine, mefloquine and halofantrine]

Arch Inst Pasteur Madagascar. 1984;51(1):81-7.
[Article in French]

Abstract

In a nine month fields study in 1983 in Madagascar, in vitro sensitivity to others drugs than 4 aminoquinolines were tested for 39 Plasmodium falciparum isolates, including 2 chloroquine resistant ones. Sensitivity to quinine, mefloquine and halofantrine were recorded from 28, 39 and 11 of these isolates respectively. IC50 with semi-microtest were under 20 nM/1 for mefloquine, under 12 nM/1 for halofantrine and under 560 nM/1 for quinine. All these values are under maximal values observed elsewhere with isolates coming from patients successfully treated with the three drugs.

Publication types

  • English Abstract

MeSH terms

  • Antimalarials / pharmacology*
  • Chloroquine / pharmacology
  • Humans
  • Mefloquine
  • Microbial Sensitivity Tests
  • Phenanthrenes / pharmacology*
  • Plasmodium falciparum / drug effects*
  • Quinine / pharmacology*
  • Quinolines / pharmacology*

Substances

  • Antimalarials
  • Phenanthrenes
  • Quinolines
  • Chloroquine
  • Quinine
  • halofantrine
  • Mefloquine