Identification of a novel integrin binding site in fibronectin. Differential utilization by beta 3 integrins

J Biol Chem. 1994 Apr 8;269(14):10856-63.

Abstract

Fibronectin (Fn) binding to the integrins alpha IIb beta 3 and alpha v beta 3 involves the Arg-Gly-Asp sequence. The identification of other regions of Fn that interact with alpha IIb beta 3 suggests a potential mechanism for differential ligand recognition by integrins. We report here the identification of an 11-residue peptide sequence from the 9th type III repeat of Fn (3Fn9), which inhibits ligand binding to alpha IIb beta 3 by interacting directly with this receptor. Mutational analysis demonstrated that this same region was involved in the formation of epitopes for two anti-Fn mAbs that inhibit Fn binding to alpha IIb beta 3, thus emphasizing the role of this site in the macromolecule. Molecular modeling of the 3Fn9-10 modules suggested that Fn residues Asp1373-Thr1383 are at least 25 A distant from the Arg-Gly-Asp site and therefore does not directly interact with it. The 3Fn9 site was differentially recognized by the beta 3 integrin family. The Asp1373-Thr1383 peptide failed to inhibit ligand binding to alpha v beta 3, a recombinant Fn Ala1235-Ser1436 fragment was not recognized by alpha v beta 3, and addition of the 3Fn9 module to the amino terminus of the 3Fn10 did not affect the potency of inhibition of Fn binding to alpha v beta 3. Thus, a novel integrin recognition site in the 3Fn9 module of Fn that is differentially recognized by the beta 3 integrins has been localized within the residues Asp1373-Thr1383.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Sequence
  • Amino Acids / metabolism
  • Antibodies, Monoclonal / immunology
  • Base Sequence
  • Binding Sites
  • DNA Primers
  • Epitopes / immunology
  • Fibronectins / immunology
  • Fibronectins / metabolism*
  • Humans
  • Integrins / metabolism*
  • Ligands
  • Models, Molecular
  • Molecular Sequence Data
  • Platelet Aggregation

Substances

  • Amino Acids
  • Antibodies, Monoclonal
  • DNA Primers
  • Epitopes
  • Fibronectins
  • Integrins
  • Ligands