Herpes simplex virus type 1 (HSV-1) uracil-DNA glycosylase: functional expression in Escherichia coli, biochemical characterization, and selective inhibition by 6-(p-n-octylanilino)uracil

Virology. 1995 Aug 1;211(1):307-11. doi: 10.1006/viro.1995.1406.

Abstract

The Herpes simplex virus type 1 (HSV-1) uracil-DNA glycosylase (UDG) is encoded by the UL2 gene. The translation from the first putative start codon of UL2 predicts a polypeptide of 334 residues, while the translation from the second start codon predicts a polypeptide of 244 residues. We have cloned and expressed the two forms of UDG, by means of the prokaryotic expression vector pMAL-c2, and both of them were enzymatically active. Furthermore, the enzymatic properties of the recombinant UDGs and of the enzyme purified from HSV-1-infected cells were similar. The two UDG polypeptides have molecular weights of 27 and 37 kDa, respectively. The 37-kDa form of recombinant UDG is consistent with the reported molecular mass of 37 kDa for the enzyme purified from HSV-1-infected cells. Both recombinant UDGs were as sensitive as UDG purified from HSV-1-infected cells to 6-(p-n-octylanilino)uracil, the most potent of a series of uracil analogs that inhibit the viral enzyme.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Base Sequence
  • Cloning, Molecular
  • Codon
  • DNA Glycosylases*
  • DNA Primers
  • DNA Repair
  • Electrophoresis, Polyacrylamide Gel
  • Escherichia coli
  • Genes, Viral
  • Herpesvirus 1, Human / enzymology*
  • Herpesvirus 1, Human / genetics
  • Kinetics
  • Molecular Sequence Data
  • Molecular Weight
  • N-Glycosyl Hydrolases / antagonists & inhibitors
  • N-Glycosyl Hydrolases / isolation & purification
  • N-Glycosyl Hydrolases / metabolism*
  • Polymerase Chain Reaction
  • Recombinant Proteins / antagonists & inhibitors
  • Recombinant Proteins / isolation & purification
  • Recombinant Proteins / metabolism
  • Restriction Mapping
  • Uracil / analogs & derivatives*
  • Uracil / pharmacology
  • Uracil-DNA Glycosidase

Substances

  • 6-(N-octylanilino)uracil
  • Codon
  • DNA Primers
  • Recombinant Proteins
  • Uracil
  • DNA Glycosylases
  • N-Glycosyl Hydrolases
  • Uracil-DNA Glycosidase

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