Platelet aggregation inhibiting and anticoagulant effects of oligoamines, XXVII. Inhibition of leucocyte adherence to endothelium by the oligoamine RE 1492C and the NO-donor RE 2047

Arch Pharm (Weinheim). 1995 Feb;328(2):125-6. doi: 10.1002/ardp.19953280206.

Abstract

The oligoamine RE 1492C (N,N',N"-4-phenylbutyl-1,3,5-benzene-trimethanamine-N,N',N"- triethylcarbamate ) inhibited the electrically provoked leucocyte adhesion to the endothelium of rat mesenteric venoles. An oral dose of 60 mg/kg gave a significant inhibition of 65-78%. This is comparable to effects seen after i.v. administration of iloprost or PGE1, respectively. In the same dosage the NO-donor RE 2047 (3-methyl-N-nitroso-sydnone-5-imine) produced an inhibition of 21-27%.

MeSH terms

  • Animals
  • Cell Adhesion / drug effects
  • Electric Stimulation
  • Endothelium, Vascular / cytology
  • Endothelium, Vascular / drug effects
  • Humans
  • In Vitro Techniques
  • Leukocytes / drug effects*
  • Platelet Aggregation Inhibitors / pharmacology*
  • Polyamines / pharmacology*
  • Rats
  • Sydnones / pharmacology*

Substances

  • 3-methylsydnone-5-nitrosimine
  • Platelet Aggregation Inhibitors
  • Polyamines
  • Sydnones
  • RE 1492