An inhibitor of protein phosphorylation stops the circadian oscillator and blocks light-induced phase shifting in Gonyaulax polyedra

J Biol Rhythms. 1994 Spring;9(1):13-26. doi: 10.1177/074873049400900102.

Abstract

The expression of circadian rhythmicity in Gonyaulax polyedra is strikingly altered by an inhibitor of protein phosphorylation. The effects of 6-dimethylaminopurine (6-DMAP), known to reversibly block cell division in many systems through inhibition of protein kinase activity, are described here for Gonyaulax. Its action appears to be exclusively tonic in nature; in cells continuously exposed, the period is lengthened in a concentration-dependent fashion. Shorter treatments at a higher concentration of 6-DMAP (5 mM) apparently stop the circadian oscillator, but reversibly so, since the rhythm resumes after drug removal with a phase delay approximately equal to the duration of the treatment. Pulses of the inhibitor are effective in causing phase delays at all times of the circadian cycle. In addition, 6-DMAP completely blocks light-induced phase advances and is effective in inhibiting many Gonyaulax protein kinases in vitro.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenine / analogs & derivatives*
  • Adenine / pharmacology
  • Animals
  • Biological Clocks / drug effects*
  • Circadian Rhythm / drug effects
  • Dinoflagellida / drug effects
  • Dinoflagellida / physiology*
  • Luminescent Measurements*
  • Phosphorylation / drug effects
  • Photoperiod
  • Protein Kinase Inhibitors
  • Protein Kinases / metabolism

Substances

  • Protein Kinase Inhibitors
  • N(6),N(6)-dimethyladenine
  • Protein Kinases
  • Adenine