Functions of the v-Src protein tyrosine kinase

Cell Biol Int. 1994 May;18(5):337-44. doi: 10.1006/cbir.1994.1083.

Abstract

The peripheral non-receptor tyrosine kinase oncoprotein, v-Src, has pleiotropic effects. It is a mitogen for quiescent cells, substituting for both competence and progression factor-mediated signals but it also induces cellular morphological transformation. We are dissecting the activities of v-Src by studying mutant proteins, including those with temperature sensitive (ts) effects, in different cellular backgrounds. Activation of a ts v-Src kinase rapidly increases activity of both the transcription factor, AP-1, and MAP kinase, an enzyme that enhances AP-1 activity by both phosphorylation of c-Jun and increased c-fos transcription; the relative contribution of these two events depends on the cells in which v-Src is expressed. Transient early AP-1 activation requires proper location of v-Src at the cell periphery and it is essential for mitogenesis. It is not, however, sufficient for entry into S-phase, there being a second need for v-Src later in G1. Transformation by v-Src does not require AP-1 activation but seems linked to events at the cell periphery, notably phosphorylation of proteins that bind to the v-Src SH3 domain such as the p85 subunit of PI-3 kinase.

Publication types

  • Review

MeSH terms

  • Animals
  • Cell Line
  • Cell Transformation, Neoplastic
  • Cells, Cultured
  • Enzyme Activation
  • Mitogen-Activated Protein Kinase 1
  • Mitosis
  • Models, Biological
  • Mutation / physiology
  • Oncogene Protein pp60(v-src) / genetics
  • Oncogene Protein pp60(v-src) / physiology*
  • Protein Serine-Threonine Kinases / metabolism
  • Protein-Tyrosine Kinases / metabolism
  • Proto-Oncogene Proteins c-jun / metabolism

Substances

  • Proto-Oncogene Proteins c-jun
  • Protein-Tyrosine Kinases
  • Oncogene Protein pp60(v-src)
  • Protein Serine-Threonine Kinases
  • Mitogen-Activated Protein Kinase 1