Intra-hippocampal injection of 8-hydroxy-2-(di-n-propylamino)tetralin (8-OH-DPAT) inhibits partial and generalized seizures induced by kindling stimulation in cats

Neurosci Lett. 1993 Sep 3;159(1-2):179-82. doi: 10.1016/0304-3940(93)90828-9.

Abstract

This study assessed the effects of microinjections of a serotonin (5-HT) 1A agonist, 8-OH-DPAT, into the feline hippocampus (HIP) on seizure response induced by electrical stimulation of this region. Intra-HIP injection of 8-OH-DPAT (10 nmol) produced a significant elevation in the afterdischarge threshold of partial HIP seizures, with a significant reduction in the duration of focal afterdischarge. Similarly, microinjection of 8-OH-DPAT at the same dose significantly raised the seizure threshold for eliciting generalized seizures in HIP-kindled cats. The present results demonstrate that focally applied 8-OH-DPAT possesses a potent anticonvulsant action, and provide further evidence for the inhibitory role of 5-HT1A receptors in the generation of HIP seizures.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 8-Hydroxy-2-(di-n-propylamino)tetralin / administration & dosage
  • 8-Hydroxy-2-(di-n-propylamino)tetralin / pharmacology*
  • Animals
  • Anticonvulsants / administration & dosage
  • Anticonvulsants / pharmacology*
  • Cats
  • Electric Stimulation
  • Electroencephalography / drug effects
  • Epilepsies, Partial / prevention & control
  • Epilepsy, Generalized / prevention & control
  • Hippocampus / physiology*
  • Kindling, Neurologic / physiology*
  • Microinjections
  • Receptors, Serotonin / drug effects
  • Receptors, Serotonin / physiology
  • Seizures / prevention & control*

Substances

  • Anticonvulsants
  • Receptors, Serotonin
  • 8-Hydroxy-2-(di-n-propylamino)tetralin