Hepatic transcriptional up-regulator of the rat microsomal epoxide hydrolase gene

DNA Cell Biol. 1994 Jan;13(1):43-50. doi: 10.1089/dna.1994.13.43.

Abstract

Rat microsomal epoxide hydrolase (mEH) is one of the detoxification enzymes and selectively expressed in liver. A 350-bp DNA fragment of the proximal promoter was found to contain information sufficient to express the mEH gene in hepatoma cells, however not in nonhepatoma cells. We identified two cis-acting elements, epoxide hydrolase proximal element 1 (EHP1) and 2 (EHP2), in this promoter region by using transient transfection assays. Each element is a new cell-type-specific transcriptional up-regulator. The cell-type-specific activity of EHP1 correlates to the limited cell distribution of its cognate transacting factor(s). In the case of EHP2, a similar or possibly the same cognate factor(s) binding to EHP2 was detected by DNase I footprinting and gel retardation assays in both hepatoma and nonhepatoma cells. However, EHP2 functions as an up-regulator only in hepatoma cells. Our finding adds repertoire to a battery of cis-regulatory elements that are required for liver-specific transcription.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Base Sequence
  • Binding Sites
  • Epoxide Hydrolases / genetics*
  • Gene Expression Regulation*
  • In Vitro Techniques
  • Microsomes, Liver / enzymology*
  • Molecular Sequence Data
  • Nuclear Proteins / metabolism
  • Oligodeoxyribonucleotides / chemistry*
  • Promoter Regions, Genetic*
  • RNA, Messenger / genetics
  • Rats
  • Transcription Factors / metabolism
  • Transcription, Genetic
  • Tumor Cells, Cultured

Substances

  • Nuclear Proteins
  • Oligodeoxyribonucleotides
  • RNA, Messenger
  • Transcription Factors
  • Epoxide Hydrolases