The TSH-dependent potassium channel in a cloned rat thyroid cell line

Biochem Biophys Res Commun. 1993 Mar 15;191(2):595-600. doi: 10.1006/bbrc.1993.1259.

Abstract

We found a TSH-dependent K+ channel in the membrane of a rat thyroid cell line (FRTL-5 cell). This K+ channel is activated by extracellular application of the thyroid stimulating hormone (TSH). Treatment of dibutyryladenosine cyclic monophosphate (Bt2 cAMP) also activated the TSH-dependent K+ channel. Intracellular application of protein kinase A activates this K+ channel without the presence of free Ca2+. These findings indicate that the thyroid K+ channel is activated through the TSH-cAMP-protein kinase A system. This is the first report of a polypeptide hormone activated K+ channel and it should be useful for examining the effects of this K+ channel on thyroid cell functions.

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Bucladesine / pharmacology
  • Calcium / metabolism
  • Clone Cells
  • Membrane Potentials
  • Molecular Sequence Data
  • Potassium Channels / drug effects*
  • Protein Kinases / metabolism
  • Rats
  • Thyroid Gland / cytology
  • Thyroid Gland / drug effects
  • Thyroid Gland / metabolism*
  • Thyrotropin / pharmacology*

Substances

  • Potassium Channels
  • Bucladesine
  • Thyrotropin
  • Protein Kinases
  • Calcium