3-Triazenopyrroles: synthesis and antineoplastic activity

Farmaco. 1993 Feb;48(2):191-4.

Abstract

Some 3-triazenopyrroles were prepared by coupling 3-diazopyrroles and secondary amines. In preliminary in vitro screening tests derivatives 3 showed to be cytotoxic and exhibited mutagenic effects.

MeSH terms

  • Animals
  • Antineoplastic Agents / chemical synthesis*
  • Antineoplastic Agents / pharmacology
  • Antineoplastic Agents / toxicity
  • Cell Survival / drug effects
  • Friend murine leukemia virus
  • Lethal Dose 50
  • Leukemia, Erythroblastic, Acute / drug therapy
  • Melanoma, Experimental / drug therapy
  • Mice
  • Mice, Inbred DBA
  • Pyrroles / chemical synthesis*
  • Pyrroles / pharmacology
  • Pyrroles / toxicity
  • Triazines / chemical synthesis*
  • Triazines / pharmacology
  • Triazines / toxicity
  • Tumor Cells, Cultured

Substances

  • Antineoplastic Agents
  • Pyrroles
  • Triazines