Alterations of striatal dopamine D2 receptors contribute to deteriorated response to L-dopa in Parkinson's disease: a [123I]-IBZM SPET study

J Neural Transm Suppl. 1995:45:113-22.

Abstract

Single photon emission tomography with the ligand [123I]-IBZM was used to image central dopamine D2 receptors in Parkinson's disease patients. The aim was to assess striatal receptor densities in relation to response to L-Dopa therapy. In the parkinsonian patients group who were untreated until SPET study and in the group of patients with a sustained response to chronic L-Dopa, striatal [123I]-IBZM uptake did not differ significantly from mean values of the control group. On the contrary, significantly diminished uptake of [123I]-IBZM was found in the basal ganglia regions of the group of patients who developed a complicated/fluctuating response to chronic L-Dopa treatment. Our results indicate that striatal D2 receptor alterations in Parkinson's disease may contribute to the altered response to L-Dopa.

MeSH terms

  • Adult
  • Aged
  • Antiparkinson Agents / pharmacology*
  • Benzamides
  • Case-Control Studies
  • Corpus Striatum / drug effects
  • Corpus Striatum / metabolism
  • Dopamine Agents / pharmacology*
  • Female
  • Humans
  • Iodine Radioisotopes
  • Levodopa / pharmacology*
  • Male
  • Middle Aged
  • Parkinson Disease / diagnostic imaging
  • Parkinson Disease / metabolism*
  • Pyrrolidines
  • Receptors, Dopamine D2 / drug effects*
  • Receptors, Dopamine D2 / metabolism
  • Tomography, Emission-Computed, Single-Photon / methods*

Substances

  • Antiparkinson Agents
  • Benzamides
  • Dopamine Agents
  • Iodine Radioisotopes
  • Pyrrolidines
  • Receptors, Dopamine D2
  • Levodopa
  • 3-iodo-2-hydroxy-6-methoxy-N-((1-ethyl-2-pyrrolidinyl)methyl)benzamide