Response of ryanodine receptor channels to Ca2+ steps produced by rapid solution exchange

Biophys J. 1996 Aug;71(2):732-41. doi: 10.1016/S0006-3495(96)79272-X.

Abstract

We used a flow method for Ca2+ activation of sheep cardiac and rabbit skeletal ryanodine receptor (RyR) channels in lipid bilayers, which activated RyRs in < 20 ms and maintained a steady [Ca2+] for 5 s. [Ca2+] was rapidly altered by flowing Ca(2+)-buffered solutions containing 100 or 200 microM Ca2+ from a perfusion tube inserted in the cis, myoplasmic chamber above the bilayer. During steps from 0.1 to 100 microM, [Ca2+] reached 0.3 microM (activation threshold) and 10 microM (maximum Po) in times consistent with predictions of a solution exchange model. Immediately following rapid RyR activation, Po was 0.67 (cardiac) and 0.45 (skeletal) at a holding voltage of +40 mV (cis/trans). Po then declined (at constant [Ca2+]) in 70% of channels (n = 25) with time constants ranging from .5 to 15 s. The mechanism for Po decline, whether it be adaptation or inactivation, was not determined in this study. cis, 2 mM Mg2+ reduced the initial Po for skeletal RyRs to 0.21 and marginally slowed the declining phase. During very rapid falls in [Ca2+] from mM (inhibited) to sub-microM (sub-activating) levels, skeletal RyR did not open. We conclude the RyR gates responsible for Ca(2+)-dependent activation and inhibition of skeletal RyRs can gate independently.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Calcium / metabolism
  • Calcium / pharmacology*
  • Calcium Channels / drug effects
  • Calcium Channels / physiology*
  • Cesium / pharmacology
  • Chlorides / pharmacology
  • Heart / physiology*
  • Ion Channel Gating
  • Kinetics
  • Lipid Bilayers
  • Membrane Potentials / drug effects
  • Muscle Proteins / drug effects
  • Muscle Proteins / physiology*
  • Muscle, Skeletal / physiology*
  • Organ Specificity
  • Rabbits
  • Ryanodine Receptor Calcium Release Channel
  • Sarcoplasmic Reticulum / physiology
  • Sheep
  • Solutions

Substances

  • Calcium Channels
  • Chlorides
  • Lipid Bilayers
  • Muscle Proteins
  • Ryanodine Receptor Calcium Release Channel
  • Solutions
  • Cesium
  • cesium chloride
  • Calcium