Roles of the N and C terminal domains of the interleukin-3 receptor alpha chain in receptor function

Blood. 1997 Feb 1;89(3):842-52.

Abstract

The interleukin-3 (IL-3), granulocyte-macrophage colony-stimulating factor, and IL-5 receptor alpha chains are each composed of three extracellular domains, a transmembrane domain and a short intracellular region. Domains 2 and 3 constitute the cytokine receptor module (CRM), typical of the cytokine receptor superfamily; however, the function of the N-terminal domain is not known. We have investigated the functions of the N-terminal and C-terminal domains of the IL-3 receptor (IL-3R) alpha chain. We find that cells transfected with the receptor beta chain (h beta c) and a truncated IL-3R alpha that is devoid of the intracellular region fail to proliferate or to activate STAT5 in response to human IL-3, despite binding the IL-3 with affinity indistinguishable from that of full-length receptor. In addition, IL-3-induced phosphorylation of h beta c was not detected. Thus, the IL-3R alpha intracellular region does not contribute detectably to stabilization of the receptor/ligand complex, but is essential for signal propagation. In contrast, a truncated IL-3R alpha with the N-terminal domain deleted interacts functionally with the beta chain; mouse cells transfected with these receptor chains proliferate in response to human IL-3 and STAT5 transcription factor is activated. High- and low-affinity binding sites are retained, although the affinity for IL-3 is decreased 15-fold, indicating a significant role for the N-terminal domain in IL-3 binding.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antibodies, Blocking / pharmacology
  • Antibodies, Monoclonal / pharmacology
  • COS Cells
  • Cytoplasm / chemistry
  • Cytoplasm / physiology
  • Intracellular Fluid / chemistry
  • Intracellular Fluid / physiology
  • Mutagenesis
  • Protein Binding
  • Protein Structure, Tertiary*
  • Receptors, Interleukin-3 / chemistry*
  • Receptors, Interleukin-3 / genetics
  • Receptors, Interleukin-3 / immunology
  • Receptors, Interleukin-3 / physiology*
  • Signal Transduction

Substances

  • Antibodies, Blocking
  • Antibodies, Monoclonal
  • Receptors, Interleukin-3