Thiazide diuretics normalize urinary calcium in spontaneously hypertensive male rats

Kidney Int. 1997 Apr;51(4):1018-21. doi: 10.1038/ki.1997.142.

Abstract

The role of the thiazide-sensitive distal convoluted tubule (DCT) in the hypercalciuria of the spontaneously hypertensive rat (SHR) strain was examined by determining (a) the renal density of the thiazide diuretic receptor with 3H-metolazone, and (b) the renal response to a maximal dose of bendroflumethiazide (BFTZ). We confirm that the renal thiazide receptor density was greater in SHR than WKY (0.936 +/- 0.026 vs. 0.797 +/- 0.045 pmol/mg protein; P = 0.02). Prior to BFTZ the urinary excretion of calcium (0.525 +/- 0.061 vs. 0.274 +/- 0.049 micromol per micromol creatinine, P < 0.01) and sodium (12.6 +/- 1.27 vs. 7.89 +/- 0.926 micromol per micromol creatinine; P < 0.01) were greater in SHR versus WKY. BFTZ decreased the excretion of calcium only in SHR and to a level (0.250 +/- 0.032) not significantly different (P = 0.519) from WKY (0.225 +/- 0.032). Surprisingly, BFTZ increased chloride excretion to a greater extent in WKY than in SHR (P = 0.008). We postulate that hypercalciuria in SHR is a manifestation of incomplete uptake of calcium from the tubule lumen across the apical cell membrane in the DCT of the SHR nephron.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Bendroflumethiazide / pharmacology*
  • Calcium / urine*
  • Chlorides / urine
  • Diuretics
  • Hypertension / drug therapy*
  • Hypertension / metabolism
  • Hypertension / urine*
  • Ion Transport / drug effects
  • Kidney Tubules, Distal / drug effects
  • Kidney Tubules, Distal / metabolism
  • Male
  • Rats
  • Rats, Inbred SHR
  • Rats, Inbred WKY
  • Sodium Chloride Symporter Inhibitors / pharmacology*

Substances

  • Chlorides
  • Diuretics
  • Sodium Chloride Symporter Inhibitors
  • Bendroflumethiazide
  • Calcium