Discriminative stimulus properties of ethanol in the rat: effects of neurosteroids and picrotoxin

Brain Res. 1997 Apr 11;753(2):348-52. doi: 10.1016/s0006-8993(97)00165-0.

Abstract

Tetrahydrodeoxycorticosterone (5beta-THDOC; 1.3-12.0 mg/kg), a neurosteroid enhancing the GABA(A) receptor-associated chloride conductance, produced predominantly ethanol-appropriate responding (> 80%) in rats trained to discriminate 1.0 g/kg ethanol from saline. However, neither picrotoxin (0.25-1.5 mg/kg), nor dehydroepiandrosterone sulfate (0.01-100.0 mg/kg), a neurosteroid acting as a GABA(A) receptor antagonist, attenuated the stimulus effects of ethanol. These results indicate that: (1) at least certain neurosteroids may produce subjective states similar to these induced by ethanol; (2) blockade of the GABA(A) receptor-associated channel does not eliminate the ethanol interoceptive cue in rats.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Dehydroepiandrosterone Sulfate / pharmacology*
  • Discrimination, Psychological*
  • Ethanol / pharmacology*
  • GABA Antagonists / pharmacology
  • Male
  • Picrotoxin / pharmacology*
  • Rats
  • Rats, Wistar
  • Sodium Chloride / pharmacology
  • Stimulation, Chemical

Substances

  • GABA Antagonists
  • Picrotoxin
  • Ethanol
  • Sodium Chloride
  • Dehydroepiandrosterone Sulfate