Effect of hydrocortisone, methylprednisolone aceponate and momethasone furoate on collagen synthesis in human skin in vivo

Skin Pharmacol. 1997;10(5-6):261-4. doi: 10.1159/000211513.

Abstract

Background: Topical corticoids decrease de novo collagen synthesis in the human skin.

Objective: We studied the effect of three corticoids, hydrocortisone (HC), methylprednisolone aceponate (MPA) and momethasone furoate (MMF) on the de novo synthesis of type I and III collagens.

Methods: Fifteen healthy male volunteers treated four areas marked on their abdominal skin for 1 week. HC was applied twice a day, MPA and MMF once a day plus vehicle once a day and vehicle twice a day. After the treatment, suction blisters were induced on the treated areas, the suction blister fluid (SBF) was collected and procollagen propeptides of type I and III procollagens (PINP, PIIINP, respectively) were analyzed by radioimmunological assays. The protein concentration in SBF was determined by a colorimetric method.

Results: All the corticoids studied decreased the procollagen propeptide concentrations in SBF. HC decreased PINP concentration by 66%, MPA by 68% and MMF by 72%. HC decreased PIIINP by 62%, MPA by 68% and MMF by 72%. The protein concentration in SBF was decreased by 11-15% by these topical corticoids.

Conclusion: HC decreases the concentration of procollagen propeptides in human skin in males to nearly the same extent as MPA and MMF.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Topical
  • Adult
  • Anti-Inflammatory Agents / pharmacology*
  • Collagen / biosynthesis*
  • Humans
  • Hydrocortisone / pharmacology*
  • Male
  • Methylprednisolone / analogs & derivatives*
  • Methylprednisolone / pharmacology
  • Mometasone Furoate
  • Peptide Fragments / metabolism
  • Pregnadienediols / pharmacology*
  • Procollagen / metabolism
  • Skin / drug effects*
  • Skin / metabolism*

Substances

  • Anti-Inflammatory Agents
  • Peptide Fragments
  • Pregnadienediols
  • Procollagen
  • procollagen Type I N-terminal peptide
  • procollagen Type III-N-terminal peptide
  • Mometasone Furoate
  • Collagen
  • methylprednisolone aceponate
  • Hydrocortisone
  • Methylprednisolone