Defects in the ubiquitin pathway induce caspase-independent apoptosis blocked by Bcl-2

J Biol Chem. 1998 Mar 13;273(11):6121-31. doi: 10.1074/jbc.273.11.6121.

Abstract

Apoptosis requires the activation of caspases (formerly interleukin 1beta-converting enzyme-like proteases), in particular those related to the caspase-3/7/6 subfamily. Recent data, however, revealed that, although caspase-specific inhibitors delay apoptosis, they are often incapable of preventing it. To obtain evidence for caspase-independent steps of apoptosis, we artificially created a high amount of short-lived or aberrant proteins by blocking the ubiquitin degradation pathway. A temperature-sensitive defect in the ubiquitin-activating enzyme E1 induced apoptosis independent of the activation of caspase-3 and -6 and the cleavage of their respective substrates poly(ADP-ribose) polymerase and lamin A. In addition, neither the caspase 3/7-specific inhibitor N-benzyloxycarbonyl-Asp-Glu-Val-Asp-fluoromethylketone nor the general caspase inhibitor N-benzyloxycarbonyl-Val-Ala-Asp-fluoromethylketone were capable of blocking this type of cell death. By contrast, Bcl-2 overexpression effectively protected cells from apoptosis induced by a defect in the E1 enzyme at the nonpermissive temperature. Bcl-2 acted downstream of the accumulation of short-lived or aberrant proteins because it did not prevent the overexpression of the short-lived proteins p53, p27(kip1), and cyclins D1 and B1 under conditions of decreased ubiquitination. These results suggest the existence of short-lived proteins that may serve the role of caspase-independent effectors of apoptosis and attractive targets of the death-protective action of Bcl-2.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amino Acid Chloromethyl Ketones / pharmacology
  • Animals
  • Apoptosis*
  • Caspase 3
  • Caspase 7
  • Caspases*
  • Cell Cycle
  • Cell Cycle Proteins*
  • Cell Line
  • Cell Nucleus / pathology
  • Cyclin B / metabolism
  • Cyclin B1
  • Cyclin D1 / metabolism
  • Cyclin-Dependent Kinase Inhibitor p27
  • Cycloheximide / pharmacology
  • Cysteine Endopeptidases / metabolism
  • Cysteine Proteinase Inhibitors / pharmacology
  • Ligases / deficiency*
  • Ligases / genetics
  • Mice
  • Microtubule-Associated Proteins / metabolism
  • Multienzyme Complexes / metabolism
  • Proteasome Endopeptidase Complex
  • Proto-Oncogene Proteins c-bcl-2 / metabolism*
  • Tumor Suppressor Protein p53 / metabolism
  • Tumor Suppressor Proteins*
  • Ubiquitin-Activating Enzymes
  • Ubiquitin-Protein Ligases

Substances

  • Amino Acid Chloromethyl Ketones
  • Ccnb1 protein, mouse
  • Cdkn1b protein, mouse
  • Cell Cycle Proteins
  • Cyclin B
  • Cyclin B1
  • Cysteine Proteinase Inhibitors
  • Microtubule-Associated Proteins
  • Multienzyme Complexes
  • Proto-Oncogene Proteins c-bcl-2
  • Tumor Suppressor Protein p53
  • Tumor Suppressor Proteins
  • benzyloxycarbonylvalyl-alanyl-aspartyl fluoromethyl ketone
  • Cyclin D1
  • Cyclin-Dependent Kinase Inhibitor p27
  • Cycloheximide
  • Ubiquitin-Protein Ligases
  • Casp3 protein, mouse
  • Casp7 protein, mouse
  • Caspase 3
  • Caspase 7
  • Caspases
  • Cysteine Endopeptidases
  • Proteasome Endopeptidase Complex
  • Ligases
  • Ubiquitin-Activating Enzymes