A 361 base pair region of the rat FSH-beta promoter contains multiple progesterone receptor-binding sequences and confers progesterone responsiveness

Mol Cell Endocrinol. 1997 Dec 31;136(1):67-78. doi: 10.1016/s0303-7207(97)00216-5.

Abstract

The rat is frequently used as a model to study the role of progesterone (P) in regulating FSH secretion and synthesis. The ability of P to modulate rat FSH-beta mRNA levels suggests the presence of a functional hormone response element. We have found three PRE-like sequences upstream of the transcription start site in the rat FSH-beta gene. These sequences are herein referred to as PRE-like sequence #1, #2 and #3 with #1 being most distal from the start site. The current studies determined whether these PRE-like sequences bound P receptor (PR) and were functional in regulating the induction of expression by P. Electrophoretic mobility shift assays (EMSA) demonstrated that a single 289 base pair (bp) DNA fragment encompassing all three PRE-like sequences specifically bound PR. Further, PR bound with high affinity to double-stranded oligonucleotides representing individual PRE-like sequences #1, #2 and, with lower affinity to a double-stranded oligonucleotide representing PRE-like sequence, #3. We have cloned a 361 bp sequence from the promoter region of the rat FSH-beta gene encompassing all three PRE-like sequences into a luciferase reporter vector (pGL3-promoter) yielding pFSHbeta361-luc+ which when transiently transfected into primary rat pituitary cell cultures, conferred P-responsiveness to a heterologous promoter. P-responsiveness was dependent upon the presence of PR and was blocked by the PR antagonist RU-486. These data strongly suggest the presence of functional PRE's in the rat FSH-beta gene promoter.

MeSH terms

  • Animals
  • Base Sequence
  • Binding Sites
  • Cells, Cultured
  • Cloning, Molecular
  • DNA / metabolism
  • Female
  • Follicle Stimulating Hormone / genetics*
  • Follicle Stimulating Hormone, beta Subunit
  • Gene Expression Regulation / genetics*
  • High Mobility Group Proteins / pharmacology
  • Humans
  • Mifepristone / pharmacology
  • Molecular Sequence Data
  • Pituitary Gland, Anterior / cytology
  • Progesterone / antagonists & inhibitors
  • Progesterone / pharmacology*
  • Progesterone Congeners / pharmacology
  • Promegestone / pharmacology
  • Promoter Regions, Genetic / genetics*
  • Rats
  • Receptors, Progesterone / metabolism*
  • Recombinant Fusion Proteins
  • Transfection

Substances

  • Follicle Stimulating Hormone, beta Subunit
  • High Mobility Group Proteins
  • Progesterone Congeners
  • Receptors, Progesterone
  • Recombinant Fusion Proteins
  • Mifepristone
  • Progesterone
  • Follicle Stimulating Hormone
  • DNA
  • Promegestone