Two distinct effectors of the small GTPase Rab5 cooperate in endocytic membrane fusion

EMBO J. 1998 Apr 1;17(7):1930-40. doi: 10.1093/emboj/17.7.1930.

Abstract

Using the yeast two-hybrid system, we have identified a novel 62 kDa coiled-coil protein that specifically interacts with the GTP-bound form of Rab5, a small GTPase that regulates membrane traffic in the early endocytic pathway. This protein shares 42% sequence identity with Rabaptin-5, a previously identified effector of Rab5, and we therefore named it Rabaptin-5beta. Like Rabaptin-5, Rabaptin-5beta displays heptad repeats characteristic of coiled-coil proteins and is recruited on the endosomal membrane by Rab5 in a GTP-dependent manner. However, Rabaptin-5beta has features that distinguish it from Rabaptin-5. The relative expression levels of the two proteins varies in different cell types. Rabaptin-5beta does not heterodimerize with Rabaptin-5, and forms a distinct complex with Rabex-5, the GDP/GTP exchange factor for Rab5. Immunodepletion of the Rabaptin-5beta complex from cytosol only partially inhibits early endosome fusion in vitro, whereas the additional depletion of the Rabaptin-5 complex has a stronger inhibitory effect. Fusion activity can mostly be recovered by addition of the Rabaptin-5 complex alone, but maximal fusion efficiency requires the presence of both Rabaptin-5 and Rabaptin-5beta complexes. Our results suggest that Rab5 binds to at least two distinct effectors which cooperate for optimal endocytic membrane docking and fusion.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Carrier Proteins / analysis
  • Carrier Proteins / genetics
  • Carrier Proteins / metabolism*
  • Cell-Free System
  • Cloning, Molecular / methods
  • Cytosol / chemistry
  • Dimerization
  • Endosomes / chemistry
  • Endosomes / metabolism*
  • GTP Phosphohydrolases / metabolism*
  • GTP-Binding Proteins / metabolism*
  • Guanine Nucleotide Exchange Factors*
  • HeLa Cells
  • Humans
  • Membrane Fusion / physiology*
  • Membrane Proteins / analysis
  • Membrane Proteins / genetics
  • Membrane Proteins / metabolism*
  • Mice
  • Molecular Sequence Data
  • Recombinant Fusion Proteins
  • Sequence Homology, Amino Acid
  • Species Specificity
  • Vesicular Transport Proteins*
  • Yeasts / genetics
  • rab5 GTP-Binding Proteins

Substances

  • Carrier Proteins
  • Guanine Nucleotide Exchange Factors
  • Membrane Proteins
  • RABEP1 protein, human
  • RABEP2 protein, human
  • RABGEF1 protein, human
  • Rabep1 protein, mouse
  • Recombinant Fusion Proteins
  • Vesicular Transport Proteins
  • GTP Phosphohydrolases
  • GTP-Binding Proteins
  • rab5 GTP-Binding Proteins