Physical interaction between retinoic acid receptor and the oncoprotein myb inhibits retinoic acid-dependent transactivation

Proc Natl Acad Sci U S A. 1998 May 12;95(10):5539-44. doi: 10.1073/pnas.95.10.5539.

Abstract

The c-myb protooncogene is predominantly expressed in hematopoietic cells and plays a vital role in hematopoiesis. Retinoic acid (RA) is able to induce differentiation of several hematopoietic cells. This differentiation is linked to decreased c-myb expression, suggesting that retinoid receptors (RAR/RXR) may down-regulate c-myb gene expression. Furthermore, recent data indicate that RAR inhibits the function of the Myb protein itself. In addition, the Myb-Ets oncogenic fusion protein has been shown to inhibit transcriptional activation by RAR and thyroid hormone receptor. Myb-Ets also antagonizes the biological response of erythrocytic progenitor cells to RA and thyroid hormone. This prompted us to investigate a possible cross talk between RAR and Myb. Here, we demonstrate that RA inhibits the expression of the endogenous Myb target gene tom-1. Conversely, Myb functions as a potent inhibitor of RA-induced biological responses. Functional analysis of Myb mutants in transfection studies revealed that the Myb DNA-binding domain (DBD) is necessary for repression whereas the transactivation domain is dispensable. Furthermore, we show that v-Myb and RAR interact in vitro and in vivo. This interaction requires the DBD of RAR. In contrast, glutathione S-transferase-pulldown assays with v-Myb mutants indicate that the DBD and the C terminus of Myb directly interact with RAR. Our results suggest that the physical interaction between Myb and RAR may play a role in the regulation of hematopoietic gene expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 3T3 Cells
  • Animals
  • Binding Sites
  • COS Cells
  • DNA / metabolism
  • DNA-Binding Proteins / metabolism
  • Gene Expression Regulation / drug effects
  • Mice
  • Oncogene Proteins v-myb
  • Protein Binding
  • Proto-Oncogene Proteins / metabolism*
  • Proto-Oncogene Proteins c-myb
  • Receptors, Retinoic Acid / metabolism*
  • Recombinant Fusion Proteins / metabolism
  • Retinoid X Receptors
  • Retroviridae Proteins, Oncogenic / metabolism
  • Trans-Activators / metabolism*
  • Transcription Factors / metabolism
  • Transcriptional Activation* / drug effects
  • Tretinoin / metabolism*

Substances

  • DNA-Binding Proteins
  • Oncogene Proteins v-myb
  • Proto-Oncogene Proteins
  • Proto-Oncogene Proteins c-myb
  • Receptors, Retinoic Acid
  • Recombinant Fusion Proteins
  • Retinoid X Receptors
  • Retroviridae Proteins, Oncogenic
  • Trans-Activators
  • Transcription Factors
  • Tretinoin
  • DNA