The ets family member Tel binds to the Fli-1 oncoprotein and inhibits its transcriptional activity

J Biol Chem. 1998 Jul 10;273(28):17525-30. doi: 10.1074/jbc.273.28.17525.

Abstract

The tel gene, recently shown to be translocated in a spectrum of acute and chronic human leukemias, belongs to the ets family of sequence-specific transcription factors. To determine the role of Tel in normal hematopoietic development, we used the tel gene as the bait in the yeast two-hybrid system to screen a hematopoietic stem cell library. Two partners were identified: Tel binds to itself, and Tel binds to the ets family member Fli-1. In vitro and in vivo assays confirmed these interactions. In transient transfection assays, Fli-1 transactivates megakaryocytic specific promoters, and Tel inhibits this effect of Fli-1. Transactivation studies using deletion mutants of Tel, and the Tel-AML-1 fusion protein, indicate that the helix-loop-helix domain of Tel only partially inhibits transactivation and that complete inhibition requires the full-length Tel molecule, including the DNA binding domain. The Tel and Fli-1 proteins are expressed early in hematopoiesis, and the inability of Tel fusion proteins such as Tel-AML-1 to counteract Fli-1 mediated transactivation may contribute to the malignant phenotype in human leukemias where this fusion protein is present.

MeSH terms

  • Base Sequence
  • Cell Differentiation
  • DNA Primers
  • DNA-Binding Proteins / antagonists & inhibitors*
  • DNA-Binding Proteins / chemistry
  • DNA-Binding Proteins / metabolism*
  • ETS Translocation Variant 6 Protein
  • Helix-Loop-Helix Motifs
  • Hematopoietic Cell Growth Factors / pharmacology
  • Hematopoietic Stem Cells / cytology
  • Hematopoietic Stem Cells / metabolism
  • Humans
  • Open Reading Frames
  • Proto-Oncogene Protein c-fli-1
  • Proto-Oncogene Proteins c-ets
  • Proto-Oncogene Proteins*
  • Repressor Proteins*
  • Trans-Activators / antagonists & inhibitors*
  • Transcription Factors / chemistry
  • Transcription Factors / metabolism*
  • Transcriptional Activation*
  • Tumor Cells, Cultured

Substances

  • DNA Primers
  • DNA-Binding Proteins
  • Hematopoietic Cell Growth Factors
  • Proto-Oncogene Protein c-fli-1
  • Proto-Oncogene Proteins
  • Proto-Oncogene Proteins c-ets
  • Repressor Proteins
  • Trans-Activators
  • Transcription Factors